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Cat. No. Product Name Target Signaling Pathways
T2700 FTI-277 hydrochloride

FTI 277 HCl

Apoptosis; Transferase; Ras Apoptosis; GPCR/G Protein; MAPK; Metabolism
FTI-277 hydrochloride (FTI 277 HCl) 是一种法尼基转移酶FTase 抑制剂,高效 Ras CAAX 肽模拟物,可抑制H-Ras 和K-Ras 信号转导,还可抑制hepatitis delta virus 感染。
T62675 FTI-277

FTI-277 是一种法尼基转移酶 FTase 抑制剂,也是一种高效 Ras CAAX 肽模拟物。FTI-277 对 H-Ras 和 K-Ras 信号转导具有抑制作用,能够抑制 hepatitis delta virus (HDV) 感染。
T41212 FTI 277

FTI 277 is a prodrug form of FTI 276 that inhibits farnesyltransferase (FTase) (IC50 = 0.5 nM). Inhibits H-Ras and K-Ras processing in whole cells (IC50 values are 0.1 and 10μM respectively) and disrupts constitutive H-Ras-specific activation of MAPK. Causes significant antiproliferative effects in human malignant glioma cells and many other tumor cell lines.

化合物

FTI-277 hydrochloride
Cat.No: T2700
Synonym: FTI 277 HCl
Target: Apoptosis, Transferase, Ras
FTI-277
Cat.No: T62675
Synonym:
Target:
FTI 277
Cat.No: T41212
Synonym:
Target:
TargetMol Loading
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