Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4535 |
Etomoxir sodium salt
(R)-(+)-乙莫克舍钠盐,(R)-Etomoxir sodium salt,Na salt,Etomoxir |
Apoptosis; Others | Apoptosis; Others |
Etomoxir sodium salt ((R)-Etomoxir sodium salt) 是一种肉碱棕榈酰转移酶 1a (CPT-1a) 抑制剂,可以阻断脂肪酸合成。Etomoxir sodium salt 具有抗肿瘤活性。 | |||
T6633 |
Ranolazine
雷诺嗪,CVT 303,Ranexa,RS 43285-003 |
Calcium Channel; Sodium Channel | Membrane transporter/Ion channel; Metabolism |
Ranolazine (RS 43285-003) 具有抗心绞痛和抗缺血的功效,通过抑制内向钠电流的后期作用 (对INa 和IKr 的IC50值分别为 6 μM 和 12 μM) 发挥作用,而不会影响心率或血压。Ranolazine 还是脂肪酸氧化 (FAO) 的部分抑制剂。 | |||
T36076 |
Ciprofibrate impurity A
|
||
Ciprofibrate impurity A is an impurity of Ciprofibrate. Ciprofibrate is a PPARα agonist[1]. [1]. Passilly, P., et al., Phosphorylation of peroxisome proliferator-activated receptor alpha in rat Fao cells and stimulation by ciprofibrate. Biochem Pharmacol, 1999. 58(6): p. 1001-8. |