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9

抑制剂 & 化合物

5

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T15266	F16 (E)-4-(3-indolylvinyl)-N-methylpyridinium iodide	Others	Others
	F16 ((E)-4-(3-indolylvinyl)-N-methylpyridinium iodide)抑制neu-overeigning 细胞的生长和乳腺上皮的增殖。
T37995	16-phenoxy tetranor Prostaglandin F2α 16-phenoxy tetranor Prostaglandin F2α
	16-phenoxy PGF2α is a metabolically stable analog of PGF2α. It binds to the FP receptor on ovine luteal cells with much greater affinity (440%) than PGF2α.
T37936	16-phenoxy tetranor Prostaglandin F2α isopropyl ester 16-phenoxy tetranor Prostaglandin F2α isopropyl ester
	Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor. Stable, lipophilic analogs of PGF2α are used to modulate luteolysis and treat glaucoma. 16-phenoxy tetranor Prostaglandin F2α isopropyl ester (16-phenoxy tetranor PGF2α isopropyl ester) is a lipophilic analog of 16-phenoxy tetranor PGF2α. Isopropyl esters of PGs serve as prodrugs, as they are efficiently hydrolyzed in certain tissues to generate the bioactive free acid.
T37937	16-phenoxy tetranor Prostaglandin F2α methyl ester 16-phenoxy tetranor Prostaglandin F2α methyl ester
	Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor. Stable, lipophilic analogs of PGF2α are used to modulate luteolysis and treat glaucoma. 16-phenoxy tetranor Prostaglandin F2α (16-phenoxy tetranor PGF2α) is a metabolically stable form of PGF2α containing a 16-phenoxy group at the ω-terminus. It binds to the FP receptor on ovine luteal cells with much greater affinity (440%) than PGF2α. 16-phenoxy tetranor PGF2α methyl ester is a lipophilic a...
T37935	16-phenoxy tetranor Prostaglandin F2α cyclopropyl methyl amide 16-phenoxy tetranor Prostaglandin F2α cyclopropyl methyl amide
	The actions of many clinical F-series prostaglandins (PGs), including those used for estrous synchronization and for reduction of intraocular pressure (IOP), are mediated through the PGF2α (FP) receptor. 16-phenoxy tetranor Prostaglandin F2α cyclopropyl methyl amide (16-phenoxy tetranor PGF2α cyclopropyl methyl amide) is an analog of PGF2α containing a 16-phenoxy group on the lower (ω) side chain and a cyclopropyl methyl amide at the C-1 position. There are no published reports on the biological...
T61936	AChE-IN-7
	AChE-IN-7 (Compound 16) 是选择性的、有效的乙酰胆碱酯酶抑制剂，抑制eeAChE 和eeBuChE 的IC50分别为 0.045 μM 和19.68 μM。AChE-IN-7 具有较高的血脑屏障渗透性。AChE-IN-7 在体内和体外都是安全的，并显示出良好的整体药代动力学性能和高生物利用度 (F = 55.5%)。
T29062	UNC3133 UNC 3133,UNC-3133
	UNC3133 is a potent and selective Mer tyrosine kinase (MerTK) inhibitor with IC50 Mer 3.0 nM; Axl 17nM; Tyro 3.31 nM; FLT3 6.6 nM; PO Cmax = 0.023; IV T1/2 = 1.59 h, %F = 16. Mer tyrosine kinase (MerTK) is aberrantly elevated in various tumor cells and ha
T36892	4'-Acetyl Chrysomycin A
	4'-Acetyl chrysomycin A is a bacterial metabolite and derivative of chrysomycin A that has been found inStreptomycesand has antibacterial and anticancer activities.1It is active against strains of methicillin-resistantS. aureus(MRSA) and vancomycin-resistant strains ofE. faecalisandE. faecium(MICs = 0.5-2 μg/ml for all). 4'-Acetyl chrysomycin A is cytotoxic against a panel of human cancer cell lines, including doxorubicin-sensitive or -resistant cells (IC50s = 0.085-0.26 and 3.4-16 ng/ml, respec...
T35978	Benastatin A
	Benastatin A is a polyketide synthase-derived benastatin that has been found inStreptomycesand has diverse biological activities.1,2,3It inhibits glutathione S-transferase (GST; Ki= 5 μM for the rat liver enzyme).2Benastatin A is active against several bacteria, including methicillin-resistantS. aureus(MRSA; MIC = 3.12 μg/ml). It induces apoptosis and cell cycle arrest at the G1/G0phase in Colon 26 mouse colon cancer cells when used at concentrations of 20 and 16 μM, respectively.3 1.Xu, Z., Sch...

化合物

Cat.No: T15266

Synonym: (E)-4-(3-indolylvinyl)-N-methylpyridinium iodide

Target: Others

16-phenoxy tetranor Prostaglandin F2α

Cat.No: T37995

Synonym: 16-phenoxy tetranor Prostaglandin F2α

16-phenoxy tetranor Prostaglandin F2α isopropyl ester

Cat.No: T37936

Synonym: 16-phenoxy tetranor Prostaglandin F2α isopropyl ester

16-phenoxy tetranor Prostaglandin F2α methyl ester

Cat.No: T37937

Synonym: 16-phenoxy tetranor Prostaglandin F2α methyl ester

16-phenoxy tetranor Prostaglandin F2α cyclopropyl methyl amide

Cat.No: T37935

Synonym: 16-phenoxy tetranor Prostaglandin F2α cyclopropyl methyl amide

Cat.No: T61936

Cat.No: T29062

Synonym: UNC 3133,UNC-3133

4'-Acetyl Chrysomycin A

Cat.No: T36892

Cat.No: T35978

Cat. No.	Product Name	Target	Signaling Pathways
TN5957	16-Deoxysaikogenin F
	16-Deoxysaikogenin F 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5957，CAS号为 57475-62-4。
TN5989	Hemslecin D 雪胆甲素-16-乙酸酯,Cucurbitacin IIa 16-acetate,23,24-Dihydrocucurbitacin F 16,25-diacetate
	Hemslecin D 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5989，CAS号为 586960-44-3。
TMA0958	Forsythoside F 连翘酯苷F,Arenarioside,三糖苯丙素苷	Xanthine Oxidase	Metabolism
	Forsythoside F (Arenarioside) 是一种黄嘌呤氧化酶 (xanthine oxidase) 抑制剂，具有抗高尿酸活性。
T37712	Fumiquinazoline D
	Fumiquinazoline D is a fungal metabolite originally isolated from A. fumigatus that has activity against Gram-positive and Gram-negative bacteria (MICs = 8-16 μg/ml) as well as F. solani and C. albicans fungi (MICs = 32 and 64 μg/ml, respectively).
TN4411	Lappaol F	CDK; P-gp; JNK	Cell Cycle/Checkpoint; MAPK; Membrane transporter/Ion channel; Neuroscience
	1. Lappaol F has antioxidant and antiaging properties, it may promote the C. elegans longevity and stress resistance through a JNK-1-DAF-16 cascade. <br/> 2. Lappaol F has potential chemosensitizing activity, it may be candidates for developing novel adju

天然产物

16-Deoxysaikogenin F

Cat.No: TN5957

Cat.No: TN5989

Synonym: 雪胆甲素-16-乙酸酯,Cucurbitacin IIa 16-acetate,23,24-Dihydrocucurbitacin F 16,25-diacetate

Cat.No: TMA0958

Synonym: 连翘酯苷F,Arenarioside,三糖苯丙素苷

Target: Xanthine Oxidase

Fumiquinazoline D

Cat.No: T37712

Cat.No: TN4411

Target: CDK, P-gp, JNK

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