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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2226 |
Pergolide mesylate
甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Pergolide mesylate salt(LY127809) 是一种有效的,具有口服活性的多巴胺 D1和 D2受体激动剂,是一种 Ergoline 衍生物,可用于帕金森氏病和高泌乳素血症的研究。 | |||
T21340 | Pergolide | ||
Pergolide, an ergoline-based dopamine receptor agonist, is used for the treatment of Parkinson's disease, which is associated with low levels of the neurotransmitter dopamine in the brain. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13686 |
Ergolide
|
NF-κB | NF-κB |
Ergolide, 源自Inula Britannica干燥花朵提取的倍半萜内酯,有效抑制RAW 264.7巨噬细胞中可诱导型一氧化氮合酶(iNOS)和环氧化酶-2(COX-2)的表达,其机制为失活NF-κB。 |