Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T77631 |
Enpp/Carbonic anhydrase-IN-2
|
Apoptosis; PDE; Carbonic Anhydrase | Apoptosis; Metabolism |
Enpp/Carbonic anhydrase-IN-2 is a potent dual inhibitor of Enpp and carbonic anhydrase, inhibiting NPP1, NPP2, NPP3, CA-IX, CA-XII, with IC50 values of 1.13, 1.07, 0.74, 0.33, 0.68, respectively.Enpp/Carbonic anhydrase-IN-2 induced apoptosis.Enpp/Carbonic anhydrase-IN-2 has antiproliferative activity against cancer cells and low cytotoxicity against normal cells. |