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Cat. No. Product Name Target Signaling Pathways
T13166 TK216

Others; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
TK216 是一种口服有效的 E26 转录因子抑制剂,具有抗癌活性。它直接结合 EWS-FLI1 并抑制 EWS-FLI1 蛋白质相互作用,也可阻止 EWS-FLI1 与 RNA 解旋酶 A 的结合。
T4638 E260

Fer and FerT inhibitor

Fer/FerT kinase Others
E260 (Fer and FerT inhibitor) 是Fer/FerT 激酶抑制剂。
T1892 Kobe2602

Raf; Ras GPCR/G Protein; MAPK
Kobe2602 是 Ras-Raf 相互作用抑制剂,具有抗癌化疗活性。它抑制 H-Ras·GTP 与 c-Raf-1 RBD 结合的Ki 值为 149 μM。
TP2468 PNU-145156E (FCE26644)

FCE 26644,FCE26644,PNU-145156E,PNU145156E,FCE-26644,PNU 145156E

PNU-145156E (FCE26644) a novel angiogenesis inhibitor, has been shown to block circulating angiogenesis promoting growth factor in animal studies and has shown anti-tumor effects in solid tumors in mice.
T24267 Kobe2601

Kobe 2601,Kobe-2601

Kobe2601 is a Kobe0065 and Kobe02602 water-soluble analog. It displays inhibitory activity towards Ras-Raf binding.

化合物

TK216
Cat.No: T13166
Synonym:
Target: Others, DNA/RNA Synthesis
E260
Cat.No: T4638
Synonym: Fer and FerT inhibitor
Target: Fer/FerT kinase
Kobe2602
Cat.No: T1892
Synonym:
Target: Raf, Ras
PNU-145156E (FCE26644)
Cat.No: TP2468
Synonym: FCE 26644,FCE26644,PNU-145156E,PNU145156E,FCE-26644,PNU 145156E
Target:
Kobe2601
Cat.No: T24267
Synonym: Kobe 2601,Kobe-2601
Target:
TargetMol Loading
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