Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3870 |
Cyasterone
杯苋甾酮,Cyasteron |
Apoptosis; EGFR | Angiogenesis; Apoptosis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Cyasterone (Cyasteron) 是主要分离自金疮小草的一种天然 EGFR 抑制剂。它通过诱导细胞凋亡和细胞周期阻滞表现出抗增殖作用,可用于抗人类肿瘤的相关研究。 | |||
T3S0237 | Precyasterone | Others | Others |
Precyasterone 是一种天然产物,分离自 Cyathula capitata 干燥的根中。 | |||
TN3681 |
Clerosterol
|
BCL; Caspase | Apoptosis; Proteases/Proteasome |
Clerosterol as a precursor of cyasterone, isocyasterone and 29-norcyasterone in biosynthesis of phytoecdysteroids of Ajuga hairy roots. Clerosterol exerts its cytotoxic effect in A2058 human melanoma cells by caspases-dependent apoptosis. |