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Cat. No.	Product Name	Target	Signaling Pathways
TP1197	Sincalide SQ19844,辛卡利特,CCK-8,Cholecystokinin octapeptide	Others	Others
	Sincalide (CCK-8) 是一种速效的胆囊收缩素的氨基酸多肽激素类似物，可在胆囊造影术中静脉使用。它的肝胆生理作用是增加胆汁的分泌，使胆囊收缩并使 Oddi 的括约肌松弛，从而使胆汁排入十二指肠。它是一种通过注射促进胆囊收缩并帮助诊断胆囊和胰腺疾病的药物。
T2312	Loxiglumide CR-1505,氯谷胺	cholecystokinin	GPCR/G Protein
	Loxiglumide (CR-1505) 是一种缩胆囊素受体拮抗剂。
TQ0062	Nastorazepide Z-360	cholecystokinin	GPCR/G Protein
	Nastorazepide 是一种选择性的、口服有效的1,5-苯并二氮杂环衍生物胃泌素/胆囊收缩素2（CCK-2）受体拮抗剂，具有抗肿瘤的潜能。
T4579	Pentagastrin 五肽胃泌素,ICI-50123	Others; cholecystokinin	GPCR/G Protein; Others
	Pentagastrin (ICI-50123) 是一种选择性的胆囊收缩素 B(CCKB) 受体激动剂，IC50=11 nM。它能够增强胃粘膜对酸的防御机制，并保护胃粘膜免受损伤。
T14932	Ceruletide Cerulein,Caerulein,雨蛙素,FI-6934	cholecystokinin	GPCR/G Protein
	Ceruletide (Caerulein) 是一种十肽，是一种安全有效的胆囊收缩剂，是一种胆囊收缩素受体激动剂，对胆囊肌肉和胆管有直接的痉挛性作用。
T1052	Proglumide 二丙谷酰胺	cholecystokinin	GPCR/G Protein
	Proglumide (Binoside) 是一种非肽的、口服具有活性的胆囊收缩素(CCK)-A/B 受体拮抗剂。它能够选择性阻断 CCK 在中枢神经系统中的作用。它能够抑制胃分泌，具有保护胃十二指肠粘膜的能力，并表现出抗癫痫和抗氧化活性。
T27503	GV150013 GV 150013,GV-150013	cholecystokinin	GPCR/G Protein
	GV150013是一种 cholecystokinin-2 (CCK2)受体拮抗剂。
T15382	GI 181771	cholecystokinin	GPCR/G Protein
	GI 181771 是胆囊收缩素 1 受体的激动剂。 GI 181771 可用于肥胖研究。
T34123	Pranazepide FR120480,FK 480,FR-120480	cholecystokinin	GPCR/G Protein
	Pranazepide (FK 480) 是一种小分子胆囊收缩素受体拮抗剂，可用于研究消化系统疾病和胰腺炎。
T9343	N-Cbz-DL-tryptophan	cholecystokinin	GPCR/G Protein
	N-Cbz-DL-tryptophan 是一种胆囊收缩素受体拮抗剂，可消除离体心脏对 CCK-8 的反应。
T14932L1	Ceruletide Ammonium Salt Caerulein Ammonium Salt,Ceruletide Ammonium Salt（17650-98-5 Free base),FI-6934 Ammonium Salt,Cerulein Ammonium Salt	cholecystokinin	GPCR/G Protein
	Ceruletide Ammonium Salt 是一种十肽，起源于热带青蛙的皮肤，是一种有效的胆囊收缩素受体 (cholecystokinin receptor) 激动剂，也是一种安全有效的胆囊收缩剂，对胆囊肌肉和胆管有直接的痉挛性作用。Ceruletide Ammonium Salt 具有镇静活性，可用于研究慢性精神分裂症。
TP2030L1	Gastrin I (human) acetate Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate,胃膜素醋酸盐	cholecystokinin	GPCR/G Protein
	Gastrin I (human) acetate (Gastrin-17 acetate) 是在胃中产生的内源性肽，通过胆囊收缩素 2 (CCK2) 受体增加胃酸分泌。
T12404	CCK-A receptor inhibitor 1	cholecystokinin	GPCR/G Protein
	CCK-A receptor inhibitor 1 是一种有效的缩胆囊素 A (CCK-A) 受体抑制剂(IC50：340 nM）。CCK-A receptor inhibitor 1 可用于研究与消化系统相关的疾病。
T26483	A-65186 A65186
	A 65186 is a Type A Cholecystokinin (CCK) receptor antagonist.
T27664	JNJ-17156516 JNJ17156516,JNJ 17156516
	JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.
T26971	Ceclazepide
	Ceclazepide is an antagonist of cholecystokinin receptor.
T23886	Cholecystokinin (27-32)-amide Cholecystokinin (27-32)-NH2
	Cholecystokinin (27-32)-amide is a CCK receptor antagonist.
T28613	RP73870 RP 73870,RP-73870
	RP73870 is a gastrin/cholecystokinin-B receptor antagonist and H2 receptor antagonist with potent anti-ulcer activity.
T24202	Jmv 167 Jmv-167,Jmv167
	Jmv 167 is an antagonist of the Cholecystokinin receptor.
T24204	Jmv 179 Jmv-179,Jmv179
	Jmv 179 is an antagonist of the cholecystokinin receptor.
T24293	L 368935 L-368935,L368,935,L-368,935,L 368,935,L368935
	L 368935 is an antagonist of the cholecystokinin receptor.
T29502	A 70874 A-70874,A70874
	A70874 has high selectivity and potency for cholecystokinin (CCK) a receptor.
T27669	JNJ-26070109 JNJ26070109
	JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat.
T28331	PD 136450 Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189
	Cholecystokinin type B receptor antagonist PD-136,450 is a partial secretory agonist in the stomach and a full agonist in the pancreas of the rat. Gastrin (cholecystokinin type B (CCK-B)) receptor antagonists may help to elucidate the physiological role o
T28335	PD 140376 PD-140376,PD140376
	PD 140376 is a highly selective antagonist radioligand for the cholecystokinin(B)-gastrin receptor in guinea pig gastric mucosa & cerebral cortex in the peripheral and central nervous systems.
T22895	L-365260 L-365,260	Others	Others
	cholecystokinin receptor 2 (CCK2) antagonist
T13261	CCK-B Receptor Antagonist 1	Others	Others
	CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.
T15101	Devazepide L-364,718,地伐西匹,MK-329	Others	Others
	Devazepide is a competitive and orally active nonpeptide antagonist of cholecystokinin (CCK) receptor (IC50s: 81 pM, 45 pM, and 245 nM for rat pancreatic, bovine gallbladder and guinea pig brain CCK receptors, respectively).
T25552	Jmv 320 Jmv-320,Jmv320
	Jmv 320 is a highly selective gastrin receptor and cholecystokinin receptor antagonist. It is a cyclic cholecystokinin-8 analog in which positions 28 and 31 have been replaced by Lys, with their side chains bridged by a succinic moiety.
T68482	CE-326597
	CE-326597 is a potent and selective CCK1R agonist. The type 1 cholecystokinin receptor (CCK1R) has multiple physiologic roles relating to nutrient homeostasis,including mediation of postcibal satiety. The type 1 cholecystokinin (CCK) receptor (CCK1R) is a key mediator of postcibal satiety and a potential target for drugs that may be useful to prevent and/or treat obesity.
T28612	RP-72540 RPR 102681,RPR-102681,RPR102681
	RP-72540 is a cholecystokinin B receptor antagonist. RP 72540 showed selectivity factors in express of 200 for CCKA versus CCKB receptors and also had high affinity for gastrin binding sites in the stomach. Administration of RP-72540 resulted in a dose-de
T17274	YM022	CCR	Immunology/Inflammation; Microbiology/Virology
	YM022 is a highly effective and selective gastrin/cholecystokinin (CCK)-B receptor antagonist. YM022 can inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation in vivo. YM022 shows the Ki values of 68 pM and 63 nM for CCK-B and CCK-A receptor, respectively.
T14932L	Ceruletide Ammonium acetate FI-6934 Ammonium acetate,Caerulein Ammonium acetate,Ceruletide Ammonium acetate (17650-98-5 free base)	cholecystokinin	GPCR/G Protein
	Ceruletide Ammonium acetate (FI-6934 Ammonium acetate) 是一种胆囊收缩素 (CCK) 受体激动剂。它是一种安全有效的胆囊动力剂和小肠和胰腺外分泌兴奋剂。
T62039	L-365260 hemihydrate
	L-365260 hemihydrate 是选择性的、具有口服活性的非肽胃泌素和脑胆囊收缩素受体 (CCK-B) 拮抗剂，Kis 值分别为 1.9 nM 和 2.0 nM。L-365260 hemihydrate 以竞争性方式与豚鼠胃泌素和脑 CCK 受体相互作用。
T8761	[Leu15]-Gastrin I human Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2	Others	Others
	[Leu15]-Gastrin I human (Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2) 基因编码人体内的蛋白质 [Leu15]-胃泌素 I。在人类染色体中，GAST 基因定位于 17q21.2。胃窦中的 G 细胞产生 [Leu15]-胃泌素 I 的前体前胃泌素。前胃泌素经过裂解和加工产生胃泌素，它对整个胃肠道上皮细胞具有营养作用。胃泌素对消化系统的生长至关重要，并刺激壁细胞产生胃酸。胃泌素通过称为胆囊收缩素(CCK) 或 CCK-B 受体 (CCK-BR) 的 G 蛋白偶联受体发挥其功能。胃泌素的释放受到食物的刺激，尤其是蛋白质饮食，并受到非常低的 pH 值的抑制。萎缩性胃炎、幽门螺杆菌感染和长期服用质子泵抑制剂感染可能导致胃泌素过度表达。胃腺癌显示高水平的胃泌素。

化合物

Cat.No: TP1197

Synonym: SQ19844,辛卡利特,CCK-8,Cholecystokinin octapeptide

Target: Others

Cat.No: T2312

Synonym: CR-1505,氯谷胺

Target: cholecystokinin

Cat.No: TQ0062

Synonym: Z-360

Target: cholecystokinin

Cat.No: T4579

Synonym: 五肽胃泌素,ICI-50123

Target: Others, cholecystokinin

Cat.No: T14932

Synonym: Cerulein,Caerulein,雨蛙素,FI-6934

Target: cholecystokinin

Cat.No: T1052

Synonym: 二丙谷酰胺

Target: cholecystokinin

Cat.No: T27503

Synonym: GV 150013,GV-150013

Target: cholecystokinin

Cat.No: T15382

Target: cholecystokinin

Cat.No: T34123

Synonym: FR120480,FK 480,FR-120480

Target: cholecystokinin

N-Cbz-DL-tryptophan

Cat.No: T9343

Target: cholecystokinin

Ceruletide Ammonium Salt

Cat.No: T14932L1

Synonym: Caerulein Ammonium Salt,Ceruletide Ammonium Salt（17650-98-5 Free base),FI-6934 Ammonium Salt,Cerulein Ammonium Salt

Target: cholecystokinin

Gastrin I (human) acetate

Cat.No: TP2030L1

Synonym: Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate,胃膜素醋酸盐

Target: cholecystokinin

CCK-A receptor inhibitor 1

Cat.No: T12404

Target: cholecystokinin

Cat.No: T26483

Synonym: A65186

Cat.No: T27664

Synonym: JNJ17156516,JNJ 17156516

Cat.No: T26971

Cholecystokinin (27-32)-amide

Cat.No: T23886

Synonym: Cholecystokinin (27-32)-NH2

Cat.No: T28613

Synonym: RP 73870,RP-73870

Cat.No: T24202

Synonym: Jmv-167,Jmv167

Cat.No: T24204

Synonym: Jmv-179,Jmv179

Cat.No: T24293

Synonym: L-368935,L368,935,L-368,935,L 368,935,L368935

Cat.No: T29502

Synonym: A-70874,A70874

Cat.No: T27669

Synonym: JNJ26070109

Cat.No: T28331

Synonym: Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189

Cat.No: T28335

Synonym: PD-140376,PD140376

Cat.No: T22895

Synonym: L-365,260

Target: Others

CCK-B Receptor Antagonist 1

Cat.No: T13261

Target: Others

Cat.No: T15101

Synonym: L-364,718,地伐西匹,MK-329

Target: Others

Cat.No: T25552

Synonym: Jmv-320,Jmv320

Cat.No: T68482

Cat.No: T28612

Synonym: RPR 102681,RPR-102681,RPR102681

Cat.No: T17274

Target: CCR

Ceruletide Ammonium acetate

Cat.No: T14932L

Synonym: FI-6934 Ammonium acetate,Caerulein Ammonium acetate,Ceruletide Ammonium acetate (17650-98-5 free base)

Target: cholecystokinin

L-365260 hemihydrate

Cat.No: T62039

[Leu15]-Gastrin I human

Cat.No: T8761

Synonym: Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2

Target: Others

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