Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10796 |
Chlormethiazole hydrochloride
氯美噻唑盐酸盐,Clomethiazole hydrochloride |
Others | Others |
Chlormethiazole hydrochloride 是抗惊厥药。它具有神经保护作用,能够阻碍 MDMA 诱导的血清素能神经末梢退化。 | |||
T14983 |
Clomethiazole
Distraneurin,Chlormethiazole,氯美噻唑,5-(2-CHLOROETHYL)-4-METHYLTHIAZOLE |
P450; GABA Receptor | Membrane transporter/Ion channel; Metabolism; Neuroscience |
Clomethiazole (Distraneurin) 是口服GABAA 激动剂,可抑制人肝微粒体中的细胞色素 P450 异构体,CYP2A6 和 CYP2E1。它有抗惊厥作用,具有治疗惊厥性癫痫持续状态的潜力。 | |||
T27007 |
Chlormethiazole edisylate
Clomethiazole ethanedisulfonate,Clomethiazole edisylate,Heminevrin,Hemithiamine,Distraneurin |
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Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic. |