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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1408 |
Capecitabine
Xeloda,卡培他滨,Capecitibine,Capiibine,RO 09-1978 |
Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Capecitabine (Capecitibine) 是一种可口服的前药,可由胸苷磷酸化酶催化转变为其活性代谢物 Fluorouracil。 | |||
T64318 |
Capecitabine-2',3'-cyclic Carbonate
|
Others | Others |
Capecitabine-2',3'-cyclic Carbonate 是一种抗增殖化合物。 | |||
T9899 |
2'',3''-Di-O-acetyl-5''-deoxy-5-fuluro-D-cytidine
|
Others | Others |
2'',3''-Di-O-acetyl-5''-deoxy-5-fuluro-D-cytidine 是 capecitabine 的衍生物。 | |||
T9900 |
5'-Deoxy-5-fluoro-N-[(pentyloxy)carbonyl]cytidine 2',3'-diacetate
|
Others | Others |
5'-Deoxy-5-fluoro-N-[(pentyloxy)carbonyl]cytidine 2',3'-diacetate 是合成 capecitabine 的中间体。 | |||
T67964 |
Terflavoxate
|
Microtubule Associated | Cytoskeletal Signaling |
Terflavoxate 是一种新型的、具有口服活性的半合成的他汀类微管抑制剂,常与卡培他滨一起联合使用。Terflavoxate 用于癌症的研究。 | |||
T21327 |
Uridine triacetate
RG 2133 triacetate,PN-401,Tri-O-acetyluridine,PN401,RG 2133,RG-2133,PN 401,RG2133,RG2133 triacetate |
Others | Others |
Uridine triacetate (RG 2133 triacetate) 是一种具有口服活性的 Uridine 前药。Uridine triacetate 能在肠道内迅速被吸收,在循环中迅速脱乙酰,生成游离尿苷。Uridine triacetate 可用于研究 5-氟尿嘧啶 (5-FU) 和卡培他滨的毒性,或早发性心脏或中枢神经系统 (CNS) 毒性。 | |||
TNU1098 | 5’-Deoxy-5-fluoro-N4-(isopentyloxycarbonyl)cytidine | ||
Nucleoside Derivatives - 5’-Modified nucleosides; 5-Modified pyrimidine nucleosides, Fluoro-modified nucleosides; Drugs and Inhibitors; 5’-Deoxy nucleosides; Capecitabine impurity E | |||
TNU1097 |
5’-Deoxy-5-fluoro-N4-[(2-methylbutoxy)carbonyl]cytidine
|
||
Nucleoside Derivatives - 5’-Modified nucleosides; 5-Modified pyrimidine nucleosides, Fluoro-modified nucleosides; Drugs and Inhibitors; 5’-Deoxy nucleosides; Capecitabine impurity E | |||
T81594 |
Osemitamab
TST001 |
||
Osemitamab是一种针对人类claudin-18.2的IgG1单克隆抗体。它由来自人鼠嵌合体TST001的γ-1链与κ链通过二硫键连接而成的二聚体(ACI)构成。该化合物与Capecitabine和Oxaliplatin联合应用,适用于胃(G)及胃食管结合部(GEJ)癌症的研究。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7965 |
5'-Deoxy-5-fluorocytidine
|
Others | Others |
5'-Deoxy-5-fluorocytidine 是 DNA 合成抑制剂 capecitabine 的中间代谢物。 |