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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T1408 Capecitabine

Xeloda,卡培他滨,Capecitibine,Capiibine,RO 09-1978

Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Capecitabine (Capecitibine) 是一种可口服的前药,可由胸苷磷酸化酶催化转变为其活性代谢物 Fluorouracil。
T64318 Capecitabine-2',3'-cyclic Carbonate

Others Others
Capecitabine-2',3'-cyclic Carbonate 是一种抗增殖化合物。
T9899 2'',3''-Di-O-acetyl-5''-deoxy-5-fuluro-D-cytidine

Others Others
2'',3''-Di-O-acetyl-5''-deoxy-5-fuluro-D-cytidine 是 capecitabine 的衍生物。
T9900 5'-Deoxy-5-fluoro-N-[(pentyloxy)carbonyl]cytidine 2',3'-diacetate

Others Others
5'-Deoxy-5-fluoro-N-[(pentyloxy)carbonyl]cytidine 2',3'-diacetate 是合成 capecitabine 的中间体。
T67964 Terflavoxate

Microtubule Associated Cytoskeletal Signaling
Terflavoxate 是一种新型的、具有口服活性的半合成的他汀类微管抑制剂,常与卡培他滨一起联合使用。Terflavoxate 用于癌症的研究。
T21327 Uridine triacetate

RG 2133 triacetate,PN-401,Tri-O-acetyluridine,PN401,RG 2133,RG-2133,PN 401,RG2133,RG2133 triacetate

Others Others
Uridine triacetate (RG 2133 triacetate) 是一种具有口服活性的 Uridine 前药。Uridine triacetate 能在肠道内迅速被吸收,在循环中迅速脱乙酰,生成游离尿苷。Uridine triacetate 可用于研究 5-氟尿嘧啶 (5-FU) 和卡培他滨的毒性,或早发性心脏或中枢神经系统 (CNS) 毒性。
TNU1098 5’-Deoxy-5-fluoro-N4-(isopentyloxycarbonyl)cytidine

Nucleoside Derivatives - 5’-Modified nucleosides; 5-Modified pyrimidine nucleosides, Fluoro-modified nucleosides; Drugs and Inhibitors; 5’-Deoxy nucleosides; Capecitabine impurity E
TNU1097 5’-Deoxy-5-fluoro-N4-[(2-methylbutoxy)carbonyl]cytidine

Nucleoside Derivatives - 5’-Modified nucleosides; 5-Modified pyrimidine nucleosides, Fluoro-modified nucleosides; Drugs and Inhibitors; 5’-Deoxy nucleosides; Capecitabine impurity E
T81594 Osemitamab

TST001

Osemitamab是一种针对人类claudin-18.2的IgG1单克隆抗体。它由来自人鼠嵌合体TST001的γ-1链与κ链通过二硫键连接而成的二聚体(ACI)构成。该化合物与Capecitabine和Oxaliplatin联合应用,适用于胃(G)及胃食管结合部(GEJ)癌症的研究。

化合物

Capecitabine
Cat.No: T1408
Synonym: Xeloda,卡培他滨,Capecitibine,Capiibine,RO 09-1978
Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
Capecitabine-2',3'-cyclic Carbonate
Cat.No: T64318
Synonym:
Target: Others
2'',3''-Di-O-acetyl-5''-deoxy-5-fuluro-D-cytidine
Cat.No: T9899
Synonym:
Target: Others
5'-Deoxy-5-fluoro-N-[(pentyloxy)carbonyl]cytidine 2',3'-diacetate
Cat.No: T9900
Synonym:
Target: Others
Terflavoxate
Cat.No: T67964
Synonym:
Target: Microtubule Associated
Uridine triacetate
Cat.No: T21327
Synonym: RG 2133 triacetate,PN-401,Tri-O-acetyluridine,PN401,RG 2133,RG-2133,PN 401,RG2133,RG2133 triacetate
Target: Others
5’-Deoxy-5-fluoro-N4-(isopentyloxycarbonyl)cytidine
Cat.No: TNU1098
Synonym:
Target:
5’-Deoxy-5-fluoro-N4-[(2-methylbutoxy)carbonyl]cytidine
Cat.No: TNU1097
Synonym:
Target:
Osemitamab
Cat.No: T81594
Synonym: TST001
Target:
Cat. No. Product Name Target Signaling Pathways
T7965 5'-Deoxy-5-fluorocytidine

Others Others
5'-Deoxy-5-fluorocytidine 是 DNA 合成抑制剂 capecitabine 的中间代谢物。

天然产物

5'-Deoxy-5-fluorocytidine
Cat.No: T7965
Synonym:
Target: Others
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