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Search Results for " cpt 11 "

5

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T78069 RPR132595A hydrochloride

NPC hydrochloride

Drug Metabolite Metabolism
RPR132595A (NPC) hydrochloride,CPT-11的活性代谢产物,由细胞色素P-450 3A4 (CYP3A4) 催化产生,经尿液排出体外。
T38474 CL2-MMT-SN38

CL2-MMT-SN38

CL2-MMT-SN38 is a derivative of SN-38, which is a potent anticancer agent and the active metabolite of Irinotecan (CPT-11), a Topoisomerase I inhibitor.
T19553 RPR132595A

NPC

Others Others
RPR132595A is an active CPT-11 metabolite, it is generated by cytochrome P-450 3A4 (CYP3A4).
T70380 ZBH-1205

ZBH-1205 is a novel camptothecin derivative, revealing potent antitumor activities mainly through cell apoptosis pathway, being more effective than cpt-11 and sn38 at inhibiting topoismerase-1
T78711 A011

ATM/ATR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
A011,作为一种选择性的ataxia-telangiectasia mutated (ATM)抑制剂,其IC50为1.0 nM,能够在与CPT-11联合应用时,诱导Apoptosis及G2/M期细胞周期阻滞,显示出显著的抗肿瘤活性。

化合物

RPR132595A hydrochloride
Cat.No: T78069
Synonym: NPC hydrochloride
Target: Drug Metabolite
CL2-MMT-SN38
Cat.No: T38474
Synonym: CL2-MMT-SN38
Target:
RPR132595A
Cat.No: T19553
Synonym: NPC
Target: Others
ZBH-1205
Cat.No: T70380
Synonym:
Target:
A011
Cat.No: T78711
Synonym:
Target: ATM/ATR
Cat. No. Product Name Target Signaling Pathways
T6228 Irinotecan

CPT-11,Topotecin,伊立替康,(+)-Irinotecan

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan (CPT-11) 是喜树碱的衍生物,是一种 DNA 拓扑异构酶 I (Topo I) 的抑制剂。Irinotecan 通过与 Topo I 复合物结合来阻止 DNA 链的重新连接,并导致双链 DNA 断裂和细胞死亡,具有抗肿瘤活性。
T0486L Irinotecan Hydrochloride

盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan Hydrochloride (CPT-11 hydrochloride) 是喜树碱半合成衍生物的盐酸盐,是一种拓扑异构酶 I 抑制剂,可研究结肠癌和直肠癌。
T0486 Irinotecan hydrochloride trihydrate

Irinotecan HCl Trihydrate,CPT-11 HCl Trihydrate,盐酸伊立替康三水合物

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan hydrochloride trihydrate (CPT-11 HCl Trihydrate) 通过抑制拓扑异构酶 1 来防止 DNA 展开,可研究结肠癌和直肠癌。

天然产物

Irinotecan
Cat.No: T6228
Synonym: CPT-11,Topotecin,伊立替康,(+)-Irinotecan
Target: Topoisomerase, Autophagy
Irinotecan Hydrochloride
Cat.No: T0486L
Synonym: 盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride
Target: Topoisomerase, Autophagy
Irinotecan hydrochloride trihydrate
Cat.No: T0486
Synonym: Irinotecan HCl Trihydrate,CPT-11 HCl Trihydrate,盐酸伊立替康三水合物
Target: Topoisomerase, Autophagy
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