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Cat. No. Product Name Target Signaling Pathways
T6321 Tofacitinib

托法替尼,Tasocitinib,CP-690550

ROCK; Apoptosis; JAK; Src Angiogenesis; Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
Tofacitinib (Tasocitinib) 是口服小分子 Janus 激酶抑制剂,用于治疗中度至重度类风湿性关节炎。
T2398 Tofacitinib Citrate

CP-690550 citrate,柠檬酸托法替尼,枸橼酸托法替尼,Tasocitinib citrate,Tofacitinib (CP-690550) Citrate

Apoptosis; Influenza Virus; JAK; Antibacterial; Antifungal Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; Microbiology/Virology; Stem Cells
Tofacitinib Citrate (CP-690550 citrate) 是 JAK1/2/3抑制剂,IC50分别为112,20 和 1 nM。它具有抗菌,抗真菌和抗病毒活性。
T69957 Quoromycin

Quoromycin is a novel antivirulence agent against Vibrio vulnificus, inhibiting the quorum-sensing signaling pathway by controlling the DNA-binding affinity of SmcR and thus effectively alleviating the virulence of V. vulnificus in vitro and in vivo.
T70167 BP-5-087

BP-5-087 is a STAT3 inhibitor, combining with BCR-ABL1 inhibition to overcome kinase-independent resistance in chronic myeloid leukemia.

化合物

Tofacitinib
Cat.No: T6321
Synonym: 托法替尼,Tasocitinib,CP-690550
Target: ROCK, Apoptosis, JAK, Src
Tofacitinib Citrate
Cat.No: T2398
Synonym: CP-690550 citrate,柠檬酸托法替尼,枸橼酸托法替尼,Tasocitinib citrate,Tofacitinib (CP-690550) Citrate
Target: Apoptosis, Influenza Virus, JAK, Antibacterial, Antifungal
Quoromycin
Cat.No: T69957
Synonym:
Target:
BP-5-087
Cat.No: T70167
Synonym:
Target:
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