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Cat. No. Product Name Target Signaling Pathways
T2342 Raxatrigine

CNV1014802,CNV 1014802,GSK-1014802,CNV-1014802

Sodium Channel Membrane transporter/Ion channel
Raxatrigine (CNV 1014802) 是有效的钠离子通道 Nav1.7抑制剂。
T41192 CNV Dopamine

CNV Dopamine is a carboxynitroveratryl (CNV)-caged dopamine; releases dopamine upon ultraviolet light stimulation (365 nm). Induces dopaminergic currents upon photolysis in brain slices expressing wild-type or GFP-labeled D2receptors. Displays no decrease in current (rundown) with UV light flash duration of up to 100 ms. Pharmacologically inactive prior to photolysis.
T71239 CNV-2197944

CNV-2197944 is a novel, small molecule, state-dependent calcium channel blocker, designed to selectively inhibit highly active Cav2.2 channels.
T71237 SC 46944

SC 46944 is a highly potent human renin inhibitor.
T2141 Mecamylamine hydrochloride

盐酸美加明,Inversine,Mevasin

AChR Neuroscience
Mecamylamine hydrochloride (Mevasin) 是一种易穿过血脑屏障的烟碱拮抗剂,用作高血压的神经节阻滞剂,具有抗神经疾病作用。
T14992 Raxatrigine hydrochloride

GSK-1014802 hydrochloride,CNV1014802 (hydrochloride)

Others Others
Raxatrigine hydrochloride is a state-dependent sodium channel blocker and a Nav1.7 sodium channel inhibitor.
T80459 ω-Conotoxin CnVIIA

Calcium Channel Membrane transporter/Ion channel; Metabolism
ω-Conotoxin CnVIIA为含27个氨基酸的神经肽类毒素,具有N型钙电流阻滞活性。
T67746 IMS2186

Others Others
IMS2186 是一种抗脉络膜新生血管 (CNV) 试剂, 可以使癌细胞周期阻滞在 G2/M 期,由此产生抗增殖和抗血管生成作用。IMS2186 能够减少眼睛渗漏和病变细胞的数量,并且无眼内毒性。
T75156L Bevasiranib sodium

Bevasiranib sodium 是一种siRNA,可沉默产生血管内皮生长因子(VEGF)的基因。VEGF 在脉络膜新生血管形成(choroidal neo-vascularization, CNV)的发病机制中起着关键作用,而CNV 是湿性年龄相关性黄斑变性(wet age-related macular degeneration, wet AMD)的前兆。
T75156 Bevasiranib

Bevasiranib 是一种siRNA,可沉默产生血管内皮生长因子(VEGF)的基因。VEGF 在脉络膜新生血管形成(choroidal neo-vascularization, CNV)的发病机制中起着关键作用,而CNV 是湿性年龄相关性黄斑变性(wet age-related macular degeneration, wet AMD)的前兆。
T70329 SH-11037

SH-11037 is a novel potent seh inhibitor, effectively blocking key angiogenic properties of human retinal endothelial cells (hrecs), inhibiting choroidal sprouting and significantly suppressing cnv lesion volume

化合物

Raxatrigine
Cat.No: T2342
Synonym: CNV1014802,CNV 1014802,GSK-1014802,CNV-1014802
Target: Sodium Channel
CNV Dopamine
Cat.No: T41192
Synonym:
Target:
CNV-2197944
Cat.No: T71239
Synonym:
Target:
SC 46944
Cat.No: T71237
Synonym:
Target:
Mecamylamine hydrochloride
Cat.No: T2141
Synonym: 盐酸美加明,Inversine,Mevasin
Target: AChR
Raxatrigine hydrochloride
Cat.No: T14992
Synonym: GSK-1014802 hydrochloride,CNV1014802 (hydrochloride)
Target: Others
ω-Conotoxin CnVIIA
Cat.No: T80459
Synonym:
Target: Calcium Channel
IMS2186
Cat.No: T67746
Synonym:
Target: Others
Bevasiranib sodium
Cat.No: T75156L
Synonym:
Target:
Bevasiranib
Cat.No: T75156
Synonym:
Target:
SH-11037
Cat.No: T70329
Synonym:
Target:
TargetMol Loading
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