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Cat. No. | Product Name | Target | Signaling Pathways |
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T3277 |
Tulobuterol hydrochloride
Lobuterol,Hokunalin,Berachin,盐酸妥布特罗 |
Influenza Virus; Adrenergic Receptor; Antibiotic | GPCR/G Protein; Microbiology/Virology; Neuroscience |
Tulobuterol hydrochloride (Hokunalin) 是一种长效的 β2肾上腺素受体激动剂,可减少慢性阻塞性肺疾病和支气管哮喘的发作频率。它也是一种拟交感神经药,用作透皮贴剂,可增加正常的横膈膜肌肉力量。它抑制鼻病毒复制并调节气道炎症。 | |||
T124293 |
Citreoviridin-C
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Citreoviridin-C 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124293,CAS号为 74145-78-1。 | |||
T80367 |
Maximin 78
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Maximin 78为一种具有广谱抗菌性能的肽类化合物。该化合物展现出针对C. albicans、S. aureus、B. subtilis的显著抗菌活性,最小抑菌浓度(MIC)分别为37.5、4.7、37.5 μg/mL。此外,Maximin 78对人类和兔子红细胞显示出溶血活性。 | |||
T124299 | Brefeldin-C | ||
Brefeldin-C 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124299,CAS号为 73899-78-2。 | |||
T67794 |
C-AFG
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C-AFG 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67794,CAS号为 110312-78-2。 | |||
T83911 |
CYY292
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CYY292是一种针对PDGFRα、PDGFRβ、FGFR1、-2和-3的抑制剂(IC50分别为5.35、4.6、28、28和78 nM)。该化合物对这些激酶的选择性高于FGFR4(IC50 > 1,000 nM),但也能抑制c-Kit、VEGFR2、VEGFR1和胰岛素样生长因子1受体(IGF-1R;IC50分别为67、33、36和75 nM),以及EGFR、布鲁顿酪氨酸激酶(BTK)、细胞周期依赖性激酶4(Cdk4)/cyclin D3和MET(IC50分别为128、198、214和396 nM)。CYY292抑制MG-63、U2OS、MNNG/HOS和Saos-2骨肉瘤细胞的增殖(IC50分别为0.84、0.76、1.36和0.72 µM)。在0.3和0.5 µM的浓度下,它抑制U87MG和LN-229胶质母细胞瘤细胞的迁移和侵袭。CYY292(30 mg/kg)在U87MG原位小鼠异种移植模型中降低肿瘤体积并增加生存率。 | |||
T36673 | CC 401 dihydrochloride | ||
High affinity JNK inhibitor (Ki values are 25-50 nM). Inhibits JNK via competitive binding of the ATP-binding site of active, phosphorylated JNK. Exhibits > 40-fold selectivity for JNK over p38, ERK, IKK2, protein kinase C, Lck and ZAP70. Hepatoprotective. Also inhibits HCMV replication. Uehara et al (2004) c-Jun N-terminal kinase mediates hepatic injury after rat liver transplantation. Transplantation. 78 324 PMID:15316358 |Uehara et al (2005) JNK mediates hepatic ischemia reperfusion injury. J... | |||
T10215 |
AAPK-25
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Apoptosis; PLK; Aurora Kinase | Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic |
AAPK-25 是选择性的Aurora/PLK 激酶双重抑制剂,显示出抗肿瘤活性。它可造成有丝分裂延迟并阻滞前中期细胞,通过生物标志物组蛋白 H3Ser10磷酸化反应,导致细胞凋亡激增。 | |||
T35683 |
2-deoxy-D-Glucose-13C6
2-deoxy-D-Glucose-13C6 |
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2-deoxy-D-Glucose-13C6is intended for use as an internal standard for the quantification of 2-deoxy-D-glucose by GC- or LC-MS. 2-deoxy-D-Glucose is a glucose antimetabolite and an inhibitor of glycolysis.1,2It inhibits hexokinase, the enzyme that converts glucose to glucose-6-phosphate, as well as phosphoglucose isomerase, the enzyme that converts glucose-6-phosphate to fructose-6-phosphate.32-deoxy-D-Glucose (16 mM) induces apoptosis in SK-BR-3 cells, as well as inhibits the growth of 143B oste... |
Cat. No. | Product Name | Target | Signaling Pathways |
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TN5812 |
Senkyunolide C
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Senkyunolide C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5812,CAS号为 91652-78-7。 | |||
TN6636 |
Formononetin-8-C-beta-D-apiofuranosyl-(1->6)-O-beta-D-glucopyranoside
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Formononetin-8-C-beta-D-apiofuranosyl-(1->6)-O-beta-D-glucopyranoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6636,CAS号为 1147858-78-3。 |