Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8326 |
BMS-2
1-(4-氟苯基)-N-[3-氟-4-(1H-吡咯并[2,3-B]吡啶-4-基氧基)苯基]-1,2-二氢-2-氧代-3-吡啶甲酰胺 |
VEGFR; FLT; c-Met/HGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
BMS-2 是 Met/Flt-3/VEGFR2 酪氨酸激酶抑制剂。 | |||
T4696 |
BMS202 hydrochloride (1675203-84-5(free base))
PD-1/PD-L1 inhibitor 2 hydrochloride |
PD-1/PD-L1 | Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation |
BMS202 hydrochloride (1675203-84-5(free base)) (PD-1/PD-L1 inhibitor 2 hydrochloride) 是一种小分子 PD-1/PD-L1 相互作用抑制剂 (IC50: 18 nM)。生物物理研究表明 BMS202 直接与 PD-L1 结合。 BMS202 的结合促进 PD-L1 二聚化并阻断 PD-L1/PD1 相互作用。 | |||
T26846 |
BMS270394
BMS 189961,BMS-270394,BMS 270394 |
||
BMS270394 is an agonist of nuclear retinoic acid receptor (RAR-γ). |