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Cat. No. Product Name Target Signaling Pathways
T6837 Flavopiridol

L868275,Alvocidib,夫拉平度,NSC 649890 HCl,HMR-1275

Apoptosis; HIV Protease; CDK; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; Microbiology/Virology; Proteases/Proteasome
Flavopiridol (Alvocidib) 是一种广谱CDK 竞争型抑制剂, 抑制 CDK1,CDK2,CDK4的IC50分别为30,170,100 nM。
T2615 Flavopiridol hydrochloride

Alvocidib Hydrochloride,NSC 649890,MDL 107826A,HL 275,FLAVOPIRIDOL HCL,NSC 649890 HCl

HIV Protease; CDK; Autophagy Autophagy; Cell Cycle/Checkpoint; Microbiology/Virology; Proteases/Proteasome
Flavopiridol hydrochloride (MDL 107826A) 是一种CDK 的广谱抑制剂,与 ATP 竞争性地抑制 CDK1,CDK2 和 CDK4 的活性,IC50值分别为 30, 170, 100 nM。
T69965 TP1287

TP-1287 is an oral phosphate prodrug of the CDK9 inhibitor, alvocidib.
T70897 Zotiraciclib HCl

Zotiraciclib, also known as TG02 and SB1317, is a novel small molecule potent CDK/JAK2/FLT3 inhibitor. Zotiraciclib may be useful for the treatment of cancer that crosses the blood brain barrier and acts by depleting Myc through the inhibition of cyclin-dependent kinase 9 (CDK9). It is one of a number of CDK inhibitors under investigation; others targeting CDK9 for the treatment of acute myeloid leukemia include alvocidib and atuveciclib. Myc overexpression is a known factor in many cancers, w...

化合物

Flavopiridol
Cat.No: T6837
Synonym: L868275,Alvocidib,夫拉平度,NSC 649890 HCl,HMR-1275
Target: Apoptosis, HIV Protease, CDK, Autophagy
Flavopiridol hydrochloride
Cat.No: T2615
Synonym: Alvocidib Hydrochloride,NSC 649890,MDL 107826A,HL 275,FLAVOPIRIDOL HCL,NSC 649890 HCl
Target: HIV Protease, CDK, Autophagy
TP1287
Cat.No: T69965
Synonym:
Target:
Zotiraciclib HCl
Cat.No: T70897
Synonym:
Target:
TargetMol Loading
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