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抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T1708 Pimobendan

Acardi,Pimobendane,UD-CG 115 BS,匹莫苯丹,UD-CG115

PDE Metabolism
Pimobendan (UD-CG 115 BS) 是一种选择性的 PDE3 抑制剂,IC50=320nM。
T35487 Anacardic Acid Diene

Anacardic acid diene is a polyunsaturated form of anacardic acid that has been found in cashew nut shell liquid. It has antibacterial activity against methicillin resistant S. aureus (MRSA) and S. mutans (MICs = 12.5 and 6.25 μg/ml, respectively). Anacardic acid diene has schistosomicidal activity against adult S. mansoni worms when used at a concentration of 100 μM. It also inhibits soybean lipoxygenase-1 in a time-dependent manner.
T126498 (15:3)-Anacardic acid

(15:3)-Anacardic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126498,CAS号为 103904-73-0。

化合物

Pimobendan
Cat.No: T1708
Synonym: Acardi,Pimobendane,UD-CG 115 BS,匹莫苯丹,UD-CG115
Target: PDE
Anacardic Acid Diene
Cat.No: T35487
Synonym:
Target:
(15:3)-Anacardic acid
Cat.No: T126498
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T6389 Anacardic Acid

漆树酸,6-pentadecylsalicylic Acid,Hydroginkgolic acid

Others; Epigenetic Reader Domain; Histone Acetyltransferase; Antibacterial Chromatin/Epigenetic; Microbiology/Virology; Others
Anacardic Acid (6-pentadecylsalicylic Acid) 是从腰果壳中提取液中分离到的酸类物质,是一种组蛋白乙酰转移酶抑制剂,对 p300 和 PCAF 的 IC50值分别为 ∼8.5 μM 和 ∼5 μM。

天然产物

Anacardic Acid
Cat.No: T6389
Synonym: 漆树酸,6-pentadecylsalicylic Acid,Hydroginkgolic acid
Target: Others, Epigenetic Reader Domain, Histone Acetyltransferase, Antibacterial
TargetMol Loading
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