Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T67836 |
AT-533
|
HSP; HSV | Cytoskeletal Signaling; Metabolism; Microbiology/Virology |
AT-533 是有效的 HSV 和 Hsp90 抑制剂。AT-533 可以阻断 HIF-1α/VEGF/VEGFR-2 信号通路,从而抑制血管生成和肿瘤生长。AT-533 也抑制下游通路的激活,包括 Erk1/2, FAK, Akt/mTOR/p70S6K。AT-533 抑制人脐静脉内皮细胞 (HUVEC) 的细胞迁移、侵袭和管形成。 | |||
T77616 |
VU533
Nape-Pld activator |
Phospholipase | Metabolism |
VU533 (Nape-Pld activator) 是一种NAPE-PLD 激活剂,其 EC50 值为0.30 µM。VU533 可以提高 NAPE-PLD 活性,增加巨噬细胞的胞葬作用。VU533 可用于与心脏代谢相关的疾病。 | |||
T38411 |
KRA-533
|
||
KRA-533, a potent KRAS agonist, directly targets the GTP/GDP binding pocket within the KRAS protein, inhibiting GTP cleavage. This inhibition leads to the buildup of constitutively active GTP-bound KRAS, which subsequently activates both apoptotic and autophagic cell death pathways specifically in cancer cells. | |||
TP2137L |
pp60 c-src (521-533) (phosphorylated) acetate
|
Others | Others |
pp60 c-src (521-533) (phosphorylated) acetate 是粘着斑形成和细胞扩散的调节剂。它还调节细胞运动,是由促运动透明质酸受体 RHAMM 触发的信号通路中的关键成分。 | |||
T71383 | NB-533 | ||
NB-533 is a macrocyclic peptidic BACE-1 inhibitor. |