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Cat. No. Product Name Target Signaling Pathways
T7683 Adenosine amine congener

ADAC

Adenosine Receptor GPCR/G Protein; Neuroscience
Adenosine amine congener (ADAC) 是一种选择性的 A1 腺苷受体激动剂,具有神经保护作用,可以改善噪音和顺铂引起的耳蜗损伤。
T5189 Omadacycline

PTK 0796,Amadacycline

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Omadacycline (Amadacycline) 是一种具有口服活性的氨基甲基环素抗菌剂,是四环素类抗生素。它与 30S 核糖体亚基结合,抑制细菌蛋白质合成。它可用于研究急性细菌性皮肤和皮肤结构感染,感染性肺炎和尿路感染。
T77018 Garadacimab

CSL312

Factor Xa Metabolism
Garadacimab (CSL312) 是有效的全人 IgG4 单克隆抗体,针对活化因子 XII (FXIIa)。Garadacimab 可用于研究遗传性血管性水肿。 。
T7503 Upadacitinib

乌帕替尼,ABT-494

JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
Upadacitinib (ABT-494) 是高效选择性的,具有口服活性的 JAK1抑制剂,IC50为43 nM,可用于多种自身免疫性疾病的研究。它对 JAK1 的选择性约为 JAK2 的 74 倍。
T20753 Omadacycline tosylate

Omadacycline tosylate is a new tetracycline.
T7503L Upadacitinib tartrate

ABT 494,ABT-494,ABT494

Upadacitinib is a potent and selective JAK inhibitor. Upadacitinib is approximately 74 fold selective for Jak1 over Jak2 in cellular assays dependent on specific, relevant cytokines. Upadacitinib demonstrates efficacy in rat arthritis models.
T68868 Hadacidin

Hadacidin is an inhibitor of AMP synthesis. Hadacidin and hadacidin analogues have anticancer activity and activity against adenylosuccinate synthetase.
T69565 Hadacidin sodium

Hadacidin sodium is an inhibitor of AMP synthesis. Hadacidin and hadacidin analogues have anticancer activity and activity against adenylosuccinate synthetase.
T71266 Omadacycline HCl

Omadacycline, also known as PTK 0796 and Amadacyclin, is a novel first-in-class aminomethylcycline with potent activity against important skin and pneumonia pathogens, including community-acquired methicillin-resistant Staphylococcus aureus (MRSA), β-hemolytic streptococci, penicillin-resistant Streptococcus pneumoniae, Haemophilus influenzae, and Legionella. Omadacycline is active against strains expressing the two main forms of tetracycline resistance (efflux and ribosomal protection). The pri...
T5189L Omadacycline mesylate

PTK 0796,PTK-0796,PTK0796

Omadacycline is an aminomethylcycline antibiotic. Omadacycline demonstrated net cidal activity in relation to the initial burden against four strains of Streptococcus pneumoniae.
T67241 SPhos Palladacycle Gen. 4

Methanesulfonato(2-dicyclohexylphosphino-2',6'-dimethoxy-1,1'-biphenyl)(2'-methylamino-1,1'-biphenyl-2-yl)palladium(II) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T67241。
T70728 Vadaclidine

Vadaclidine is an orally acting antinociceptive muscarinic agonist.

化合物

Adenosine amine congener
Cat.No: T7683
Synonym: ADAC
Target: Adenosine Receptor
Omadacycline
Cat.No: T5189
Synonym: PTK 0796,Amadacycline
Target: ribosome, Antibacterial, Antibiotic
Garadacimab
Cat.No: T77018
Synonym: CSL312
Target: Factor Xa
Upadacitinib
Cat.No: T7503
Synonym: 乌帕替尼,ABT-494
Target: JAK
Omadacycline tosylate
Cat.No: T20753
Synonym:
Target:
Upadacitinib tartrate
Cat.No: T7503L
Synonym: ABT 494,ABT-494,ABT494
Target:
Hadacidin
Cat.No: T68868
Synonym:
Target:
Hadacidin sodium
Cat.No: T69565
Synonym:
Target:
Omadacycline HCl
Cat.No: T71266
Synonym:
Target:
Omadacycline mesylate
Cat.No: T5189L
Synonym: PTK 0796,PTK-0796,PTK0796
Target:
SPhos Palladacycle Gen. 4
Cat.No: T67241
Synonym:
Target:
Vadaclidine
Cat.No: T70728
Synonym:
Target:
TargetMol Loading
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