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Cat. No. Product Name Target Signaling Pathways
T36832 PDE4B-IN-2

A 33

PDE Metabolism
PDE4B-IN-2 (A 33) 是一种具有口服活性,选择性 PDE4B 抑制剂,IC50 为 15 nM。PDE4B-IN-2 抑制 PDE4D (IC50=1.7 µM)。PDE4B-IN-2 表现出有效的抗炎作用。
T40950 A3334

A3051, is a robust and orally active inhibitor of CXXC5-DVL with an IC 50 of 63.06 nM. Its applications include research into phenotypes associated with obesity, diabetes, and NASH that are induced by high fat diet (HFD) and methionine-choline deficient diet (MCD).
T83226 A3373

Phospholipase Metabolism
A3373 是新型 PLD1 和 PLD2 抑制剂,对 PLD1 的 IC50 为 325 nM ,对 PLD2 的 IC50 为 15.15 µM,能够有效抑制 LPS 诱导的免疫反应,并在自身免疫性关节炎、骨脱矿及破骨细胞生成等方面发挥关键作用。
T68826 A33903

A33903 is a 1,4-benzodiazepine analog that is being studied as a potential inhibitor of respiratory syncytial virus. This molecule was moderately active and demonstrated good pharmacokinetic properties.
T26480 A331440

A-331440,A331440 free base,A 331440

A331440 is an modulator of L-histidine and histamine H3 receptor.
T22935 LU AA33810

Others Others
neuropeptide Y (NPY) Y5 receptor antagonist

化合物

PDE4B-IN-2
Cat.No: T36832
Synonym: A 33
Target: PDE
A3334
Cat.No: T40950
Synonym:
Target:
A3373
Cat.No: T83226
Synonym:
Target: Phospholipase
A33903
Cat.No: T68826
Synonym:
Target:
A331440
Cat.No: T26480
Synonym: A-331440,A331440 free base,A 331440
Target:
LU AA33810
Cat.No: T22935
Synonym:
Target: Others
TargetMol Loading
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