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Cat. No.	Product Name	Target	Signaling Pathways
T2344	LY 344864 LY344864	5-HT Receptor	GPCR/G Protein; Neuroscience
	LY 344864 是一种特异性受体激动剂，有对克隆 5-HT1F 受体的亲和力，Ki 为6 nM。
T4266	LY334370 4-氟-N-(3-(1-甲基哌啶-4-基)-1H-吲哚-5-基)苯甲酰胺盐酸盐,LY 334370	5-HT Receptor	GPCR/G Protein; Neuroscience
	LY334370 是一种选择性5-HT1F 受体激动剂，Ki 值为 1.6 nM。
T2344L	LY 344864 racemate	5-HT Receptor	GPCR/G Protein; Neuroscience
	LY 344864 racemate 是一种 5-HT1F 受体激动剂。
T4118	SB 271046 hydrochloride SB 271046A	5-HT Receptor	GPCR/G Protein; Neuroscience
	SB 271046 hydrochloride (SB 271046A) 是高效、选择性和具有口服活性的5-HT6受体拮抗剂，对大鼠、猪和人的pKi 分别为 9.02、8.55 和 8.81。它增加额叶皮层中的细胞外天冬氨酸和谷氨酸并表现出抗惊厥活性，EC50为 0.16 μM。它对 5-HT6 受体、结合位点和离子通道的选择性超过 200 倍。
T1092	Zolmitriptan 佐米曲普坦,311C90,BW-311C90	5-HT Receptor	GPCR/G Protein; Neuroscience
	Zolmitriptan (311C90) 是一种5-HT1B/1D 受体部分激动剂，可用于偏头痛的研究，对 5-HT1B、5-HT1D、5-HT1F 受体的Ki 分别为 5.01、0.63 和 63.09 nM。
T22952	LY 334370 hydrochloride	Others	Others
	5-HT1F receptor agonist
T11902	LY 344864 S-enantiomer	Others	Others
	LY 344864 S-enantiomer, the S-enantiomer of LY344864, serves as a 5-HT1F receptor agonist.
T27915	LY 302148 LY-302148,LY302148
	LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.
T27059	CP-122288
	CP-122288 is a potent and selective agonist for the 5-HT1B, 5-HT1D and 5-HT1F serotonin receptor subtypes. CP-122288 is potent as an inhibitor of plasma protein extravasation and neurogenic inflammation.
T19690	SB 224289 SB224289,SB-224289
	SB 224289 is a selective antagonist of 5-HT1B receptor with pKi of 8.2. It is a centrally active following oral administration in vivo. SB 224289 displays 60-fold selectivity over 5-HT1D, 5-HT1A, 5-HT1E, 5-HT1F, 5-HT2A and 5-HT2C receptors in radioligand
T41295	LY 344864 hydrochloride
	LY 344864 hydrochloride 是选择性的受体激动剂，对5-HT1F 受体具有6 nM(Ki)的亲和力。
T2459	BRL 54443 BRL54443	5-HT Receptor	GPCR/G Protein; Neuroscience
	BRL 54443 是一种有效的 5-HT1E/1F 受体激动剂，pKi 值分别为 8.7 和 8.9。