Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1445 |
Agomelatine
Thymanax,S-20098,Valdoxan,阿戈美拉汀 |
Melatonin Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Agomelatine (Valdoxan) 是褪黑激素受体的强效激动剂和 5-羟色胺-2C (5-HT2C) 受体的拮抗剂,在猪和人 5-HT2C 克隆受体中pKi 分别为 6.4 和 6.2。 | |||
T10267 |
Agomelatine (L(+)-Tartaric acid)
阿戈美拉汀 L(+)-酒石酸,S-20098 L(+)-Tartaric acid |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and HEK-hMT2). It also is a selective 5-HT2C receptor antagonist (pKis: 6.4 and 6.2 at native (porcine) and cloned (human) 5-HT2C receptors). | |||
T60523 |
Agomelatine hydrochloride
S-20098 hydrochloride |
MT Receptor | Neuroscience |
Agomelatine hydrochloride (S-20098 hydrochloride) (S-20098 hydrochloride) 是特异性的MT1和MT2受体激动剂,对 CHO-hMT1的Ki 值为0.1 nM,对HEK-hMT1的Ki 值为0.06 nM,对CHO-hMT2的Ki 值为0.12 nM,对HEK-hMT2 的Ki 值为0.27 nM。Agomelatine hydrochloride 是选择性的5-羟色胺2C(5-HT2C)受体拮抗剂,对天然 (猪) 和克隆的人 5-HT2C 受体的pKi 值分别为 6.4 和 6.2。 | |||
T10266 |
Agomelatine-d6
Agomelatine D6,S-20098 D6 |
Others | Others |
Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors. |