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Cat. No. Product Name Target Signaling Pathways
T2078 Fimepinostat

CUDC-907,PI3K/HDAC Inhibitor,CUDC 907

Apoptosis; PI3K; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Fimepinostat (CUDC 907) 是一种 I 型PI3K 及 I 和 II 型HDAC 酶抑制剂,作用于 PI3Kα/PI3Kβ/PI3Kδ 和 HDAC1/HDAC2/HDAC3/HDAC10 ,IC50分别为 19/54/39 nM 和 1.7/5.0/1.8/2.8 nM。
T70759 CUDC-907 mesylate

CUDC-907 mesylate is a small molecule inhibitor of histone deacetylase and PI3 kinase developed by Curis. It is investigated in clinical trials for the treatment of relapsed or refractory lymphomas, thyroid cancer, multiple myeloma, breast cancer and other malignancies.

化合物

Fimepinostat
Cat.No: T2078
Synonym: CUDC-907,PI3K/HDAC Inhibitor,CUDC 907
Target: Apoptosis, PI3K, HDAC
CUDC-907 mesylate
Cat.No: T70759
Synonym:
Target:
TargetMol Loading
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