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Cat. No. Product Name Target Signaling Pathways
T3455 Merestinib

LY2801653

Discoidin Domain Receptor (DDR); FLT; c-Met/HGFR; ROS; ROS Kinase Angiogenesis; Immunology/Inflammation; Tyrosine Kinase/Adaptors
Merestinib (LY2801653) 是一种有效的口服生物可利用的具有抗肿瘤活性的c-Met 抑制剂。
T15808 Merestinib dihydrochloride

LY2801653 dihydrochloride

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
Merestinib dihydrochloride is an effective and orally bioavailable c-Met inhibitor (Ki=2 nM). It has anti-tumor activities and also has potent activity against MST1R (IC50=11 nM), FLT3 (IC50=7 nM), AXL (IC50=2 nM), MERTK (IC50=10 nM), TEK (IC50=63 nM), RO

化合物

Merestinib
Cat.No: T3455
Synonym: LY2801653
Target: Discoidin Domain Receptor (DDR), FLT, c-Met/HGFR, ROS, ROS Kinase
Merestinib dihydrochloride
Cat.No: T15808
Synonym: LY2801653 dihydrochloride
Target: ROCK
TargetMol Loading
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