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Cat. No. Product Name Target Signaling Pathways
T6087 AZD 6482

KIN 193,AZD6482

DNA-PK; PI3K; Autophagy Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
AZD 6482 (AZD6482) 是一种有效的选择性p110β抑制剂,IC50为 0.69 nM。它也是 PI3Kβ 抑制剂,IC50 为 10 nM。
T12658 (Rac)-AZD 6482

(Rac)-KIN-193

Others Others
(Rac)-AZD 6482 is the racemate of AZD 6482. AZD 6482 is a potent and selective inhibitor of p110β (IC50 of 0.69 nM).
T30261 AZD6482 (S-isomer)

AZD-6482,AZD 6482,AZD6482 (S),AZD6482

AZD6482 (S-isomer) is a potent, selective, ATP-competitive PI3Kβ inhibitor (IC(50) 0.01 μm), which can inhibit insulin-induced in vitro glucose uptake by human adipocytes (IC(50) is 4.4 μm).

化合物

AZD 6482
Cat.No: T6087
Synonym: KIN 193,AZD6482
Target: DNA-PK, PI3K, Autophagy
(Rac)-AZD 6482
Cat.No: T12658
Synonym: (Rac)-KIN-193
Target: Others
AZD6482 (S-isomer)
Cat.No: T30261
Synonym: AZD-6482,AZD 6482,AZD6482 (S),AZD6482
Target:
TargetMol Loading
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