Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1119 |
Rasagiline
雷沙吉兰,AGN1135,TVP1012 |
BCL; MAO; Monoamine Oxidase | Apoptosis; Metabolism; Neuroscience |
Rasagiline (AGN1135) 是不可逆的、高效的、选择性的线粒体单胺氧化酶 (MAO) 抑制剂,抑制大鼠脑 MAO B 和 MAO A 的 IC50分别为 4.43 nM 和 412 nM。 | |||
T6962 |
Rasagiline Mesylate
TVP1012,甲磺酸雷沙吉兰,AGN1135,Azilect |
Apoptosis; MAO; Autophagy; Monoamine Oxidase | Apoptosis; Autophagy; Metabolism; Neuroscience |
Rasagiline Mesylate (AGN1135) 是一种高效的,不可逆的选择性线粒体单胺氧化酶 (MAO) 抑制剂,抑制大鼠脑 MAO B 和 MAO A 的IC50分别为 4.43 nM 和 412 nM。 | |||
T13252 |
(S)-Rasagiline
TVP1022,(S)-雷沙吉兰,S-PAI |
Others | Others |
(S)-Rasagiline is rasagiline S-isomer, and is an agent of anti-Parkinson. | |||
T13252L |
(S)-Rasagiline mesylate
TVP1022 (mesylate),(S)-雷沙吉兰甲磺酸,S-PAI mesylate |
Others | Others |
(S)-Rasagiline mesylate is rasagiline S-isomer, and is an agent of anti-Parkinson. | |||
T71910 |
Racemic rasagiline
|
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Racemic rasagiline,也称为 AGN-1135,是一种单胺氧化酶 B 型抑制剂(MAOI)。然而,在食用富含酪胺的食物的患者中,这种药物的应用可能导致致命的高血压危象。TVP-1022是雷沙吉兰的(S)异构体,具有心脏保护剂的作用。 |