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Cat. No. Product Name Target Signaling Pathways
T1291 Cisapride

西沙必利,西沙比利,Prepulsid,R 51619,Pridesia,Kaudalit,(±)-Cisaprid,Kinestase

Potassium Channel; 5-HT Receptor; HER Angiogenesis; GPCR/G Protein; JAK/STAT signaling; Membrane transporter/Ion channel; Neuroscience; Tyrosine Kinase/Adaptors
Cisapride (R 51619) 是一种5-HT4受体激动剂,还是 hERG 抑制剂。它可作用于肠道中的血清素受体,促进肠道蠕动,增加胃排空并减少食管反流。
T22296 Cisapride hydrate

Propulsid,Alimix,Enteropride,Kinestase,西沙比利,Propulsin

EGFR; 5-HT Receptor Angiogenesis; GPCR/G Protein; JAK/STAT signaling; Neuroscience; Tyrosine Kinase/Adaptors
Cisapride acts directly as a selective agonist of serotonin 5-HT4 receptor with IC50 value of 0.483 μM. And It also acts indirectly as a parasympathomimetic.

化合物

Cisapride
Cat.No: T1291
Synonym: 西沙必利,西沙比利,Prepulsid,R 51619,Pridesia,Kaudalit,(±)-Cisaprid,Kinestase
Target: Potassium Channel, 5-HT Receptor, HER
Cisapride hydrate
Cat.No: T22296
Synonym: Propulsid,Alimix,Enteropride,Kinestase,西沙比利,Propulsin
Target: EGFR, 5-HT Receptor
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