Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1549 |
Raloxifene hydrochloride
LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl |
Estrogen Receptor/ERR; Others; MAO; Estrogen/progestogen Receptor; Autophagy | Autophagy; Endocrinology/Hormones; Metabolism; Neuroscience; Others |
Raloxifene hydrochloride (LY156758 hydrochloride) 是一种选择性且可口服的雌激素受体调节剂,用于预防绝经后妇女的骨质疏松症。它对骨骼和胆固醇代谢具有雌激素激动作用,但对乳腺和子宫组织具有完全的雌激素拮抗作用。 |