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Cat. No. Product Name Target Signaling Pathways
T2318 Sacubitril/Valsartan

Sacubitril mixture with Valsartan,沙库必曲/缬沙坦,Valsartan,Sacubitril,LCZ696

Apoptosis; RAAS; Neprilysin Apoptosis; Endocrinology/Hormones; Metabolism
Sacubitril/Valsartan (LCZ696),以1:1摩尔比由Valsartan(一种ARB)和Sacubitril(AHU377)组成,为创新口服血管紧张素受体-脑啡肽酶(ARN)双重抑制剂,旨在治疗高血压与心力衰竭。其作用机制包括抑制炎症、氧化应激及细胞凋亡,有助于改善糖尿病心肌病。
T19622 (Z)2S,4R-Sacubitril

Others Others
(Z)2S,4R-Sacubitril is the impurity of Sacubitril. Sacubitril is used in combination with valsartan for the treatment of patients with heart failure.
T19114L Sacubitril-(2S,4S)-Isomer

(2S,4S)-Sacubitril,LCZ 696杂质C

Others Others
Sacubitril-(2S,4S)-Isomer ((2S,4S)-Sacubitril) 是 Sacubitril 的异构体,它是一种脑啡肽酶抑制剂。
T19114 (2S,4S)-Sacubitril

Sacubitril Impurity C,LCZ 696杂质C

Others Others
(2S,4S)-Sacubitril (Sacubitril Impurity C) 是 Sacubitril 的杂质。其中 Sacubitril 是 NEP 抑制剂,可用于研究心力衰竭。

化合物

Sacubitril/Valsartan
Cat.No: T2318
Synonym: Sacubitril mixture with Valsartan,沙库必曲/缬沙坦,Valsartan,Sacubitril,LCZ696
Target: Apoptosis, RAAS, Neprilysin
(Z)2S,4R-Sacubitril
Cat.No: T19622
Synonym:
Target: Others
Sacubitril-(2S,4S)-Isomer
Cat.No: T19114L
Synonym: (2S,4S)-Sacubitril,LCZ 696杂质C
Target: Others
(2S,4S)-Sacubitril
Cat.No: T19114
Synonym: Sacubitril Impurity C,LCZ 696杂质C
Target: Others
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