Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GLN-1062 是 galantamine 的前体药物,在阿尔兹海默症中有研究价值。
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
1 mg | ¥ 638 | 现货 | ||
5 mg | ¥ 1,570 | 现货 | ||
10 mg | ¥ 2,420 | 现货 | ||
25 mg | ¥ 3,930 | 现货 | ||
50 mg | ¥ 5,720 | 现货 | ||
100 mg | ¥ 7,750 | 现货 | ||
500 mg | ¥ 15,500 | 待询 | ||
1 mL * 10 mM (in DMSO) | ¥ 1,670 | 现货 |
产品描述 | GLN-1062 is a pro-drug of galantamine and liberates galantamine on cleavage by a carboxyesterase in the brain. |
体内活性 | GLN-1062 has more than 15-fold higher bioavailability in the brain than the same doses of galantamine. In animal models of drug-induced amnesia, GLN-1062 produced several fold larger cognitive improvement than the same doses of galantamine, without exhibiting any significant levels of gastrointestinal side effects that are typical for the unmodified drug and other inhibitors of cholinesterases, such as donepezil and rivastigmin. In the ferret, dramatically reduced emetic and behavioral responses were observed when GLN-1062 was administered instead of galantamine[1]. |
分子量 | 391.46 |
分子式 | C24H25NO4 |
CAS No. | 224169-27-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45 mg/mL (114.95 mM)
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO | 1 mM | 2.5545 mL | 12.7727 mL | 25.5454 mL | 63.8635 mL |
5 mM | 0.5109 mL | 2.5545 mL | 5.1091 mL | 12.7727 mL | |
10 mM | 0.2555 mL | 1.2773 mL | 2.5545 mL | 6.3863 mL | |
20 mM | 0.1277 mL | 0.6386 mL | 1.2773 mL | 3.1932 mL | |
50 mM | 0.0511 mL | 0.2555 mL | 0.5109 mL | 1.2773 mL | |
100 mM | 0.0255 mL | 0.1277 mL | 0.2555 mL | 0.6386 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
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