Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T79930 | Sanggenon A
桑根酮A
|
76464-71-6 | 98% |
|
Sanggenon A通过调控BV2和RAW264.7细胞中的NF-κB及HO-1/Nrf2信号途径,展现了抗炎效果。该化合物明显抑制了由脂多糖(LPS)引起的一氧化氮产生。 | ||||
T79932 | Eudebeiolide B
化合物 Eudebeiolide B
|
1934299-51-0 | 98% |
|
Eudebeiolide B,一种自荔枝草分离得的化合物,能通过调控RANKL诱导的NF-κB、c-Fos及钙信号来抑制破骨细胞的生成,适用于研究与破骨细胞相关的疾病。 | ||||
T79933 | (−)-N-Hydroxyapiosporamide
化合物 (−)-N-Hydroxyapiosporamide
|
1205676-02-3 | 98% |
|
(−)-N-Hydroxyapiosporamide (NHAP)为生物碱类NF-κB抑制剂,表现出体外及体内抗肿瘤活性,常用于结直肠癌(CRC)研究。 | ||||
T79999 | NF-κB-IN-13
化合物 NF-κB-IN-13
|
117596-92-6 | 98% |
|
NF-κB-IN-13(compound 12)在RAW264.7巨噬细胞中显著抑制了LPS诱导的NF-κB激活以及NO生成,表现出其抗炎效果。 | ||||
T80062 | Mitogen-activated protein kinase 1
化合物 Mitogen-activated protein kinase 1
|
137632-08-7 | 98% |
|
Mitogen-activated protein kinase1 (MAPK1) 能够激活下游的 p38/NF-κB 通路,并调控多种与脓毒症相关的疾病细胞过程。此外,MAPK1 通过磷酸化催化底物蛋白,起到调节底物蛋白活性开关的作用。 | ||||
T80208 | Tripeptide-41
化合物 Tripeptide-41
|
1093241-16-7 | 98% |
|
Tripeptide-41(CG-Lipoxyn)作为一种生物活性肽,具备降低脂肪积聚的功能,常见于化妆品成分应用。 | ||||
T82022 | IVMT-Rx-3
化合物 IVMT-Rx-3
|
98% |
|
|
IVMT-Rx-3是针对SDCBP的PDZ1和PDZ2结构域,特别是MDA-9/Syntenin的抑制剂。该化合物能够中断MDA-9/Syntenin与Src之间的互动,减少NF-κB的激活,并且降低MMP-2/MMP-9的表达量,从而抑制了黑色素瘤的转移。 | ||||
T82049 | IR-Crizotinib
化合物 IR-Crizotinib
|
2387927-74-2 | 98% |
|
IR-Crizotinib是一种结合了近红外染料IR-786和Crizotinib的复合物,能穿透血脑屏障及在小鼠颅内荧光定位GBM。作为NIK抑制剂,其IC50值为3.381 μM,既能有效抑制胶质瘤细胞体外生长及侵袭,也适用于体内研究,对癌症治疗具有研究意义。 | ||||
T82665 | CTP-NBD
化合物 CTP-NBD
|
1268513-27-4 | 98% |
|
CTP-NBD (CTP-NBD) 是一种具有细胞渗透性的特异性 NFκB (NFκB) 抑制剂,常用于结肠炎研究。 | ||||
T83052 | Anti-inflammatory agent 60
化合物 Anti-inflammatory agent 60
|
98% |
|
|
Anti-inflammatory agent 60 (compound 21) 的 IC50 值针对一氧化氮生成为 12.95 μM。此化合物通过浓度依赖性方式降低 iNOS、phosphorylated p65 以及 β-catenin 的表达。 | ||||
TN4038 | Eupatolide
泽兰内酯
|
6750-25-0 | 98% |
|
Eupatolide 是从 Inula japonica 的花中分离出来的,具有抗炎活性。 Eupatolide 可用于研究乳腺癌细胞对 TRAIL 的耐药性。 | ||||
TN3587 | Capillarisin
化合物 TN3587
|
56365-38-9 | 98% |
|
Capillarisin is a novel blocker of STAT3 activation and thus may have a potential in negative regulation of growth, metastasis, and chemoresistance of tumor cell... | ||||
TN1806 | Isotetrandrine
异汉防己甲素
|
477-57-6 | 98% |
|
Isotetrandrine is a small molecule inhibitor, on various aspects of LPS-induced inflammation in vitro and in vivo. It dose-dependently suppresses the severity of... | ||||
TN1485 | Chicanine
襄五脂素
|
78919-28-5 | 98% |
|
Chicanine has anti-inflammatory activity in macrophages by down-regulating LPS-induced inflammatory cytokines in IκBα±/MAPK/ERK signaling pathways. | ||||
TN2095 | Pomiferin
橙桑黄酮
|
572-03-2 | 98% |
|
Pomiferin is a natural product inhibitor of carbonic anhydrase I and II isoenzymes. It has anticancer, antibacterial and antidiabetic properties. Pomiferin has a... | ||||
TMA1777 | Hydrangenol 8-O-glucoside
化合物 TMA1777
|
67600-94-6 | 98% |
|
Hydrangenol 8-O-glucoside may have anti-inflammary activity. | ||||
TN3410 | Anatabine
化合物 TN3410
|
581-49-7 | 98% |
|
Anatabine shows anti-inflammatory activity in vitro and in vivo, which is mediated in part via an inhibition of STAT3 phosphorylation.Anatabine has anti-Alzheime... | ||||
TN4633 | Neocryptotanshinone II
化合物 TN4633
|
27468-20-8 | 98% |
|
Neocryptotanshinone inhibits lipopolysaccharide-induced inflammation in RAW264.7 macrophages by suppression of NF-κB and iNOS signaling pathways. | ||||
TN4263 | Isoangustone A
化合物 TN4263
|
129280-34-8 | 98% |
|
Isoangustone A has antitumor activity, it can induce G1 cycle arrest in DU145 human prostate and 4T1 murine mammary cancer cells, it inhibits cell proliferation ... | ||||
T4366 | Quinovic acid
化合物 T4366
|
465-74-7 | 98% |
|
Quinovic acid shows some anti-tumour activities, quinovic acid glycosides have a potent inhibitory effect on the growth of human bladder cancer cell lines by ind... |