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抑制剂 & 化合物

4

天然产物

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Cat. No. Product Name Target Signaling Pathways
T30002 Ammifurin

Ammifurin is a Furocoumarin mixture used in treatment of vitiligo.

化合物

Ammifurin
Cat.No: T30002
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0759 Monobenzone

4-苄氧基苯酚,Benoquin

Tyrosinase Proteases/Proteasome
Monobenzone (Benoquin) 是皮肤脱色剂。它可引起色素脱失和活跃的人白癜风,对白癜风具有潜在的研究价值。
T1431 Khellin

凯林,Amicardine,Methafrone,Visammin

EGFR; Others Angiogenesis; JAK/STAT signaling; Others; Tyrosine Kinase/Adaptors
Khellin (Methafrone) 是从阿米芹中提取得到的一种呋喃并色酮,是EGFR 抑制剂,IC50为 0.15 µM。它体外具有抗增殖活性,还具有抗痉挛和冠状动脉舒张作用。
T4558 Trioxsalen

三甲沙林,Trimethylpsoralen,Trioxysalen,Trisoralen

DNA Alkylator/Crosslinker; DHFR Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Trioxsalen (Trioxysalen) 是一种呋喃香豆素和补骨脂素衍生物,与 UV-A 一起用于光疗治疗白癜风和手部湿疹。它是一种光化学 DNA 交联剂,可用于激光激活定位的基因组链间交联可视化。
T40859 5-Hydroxy-8-methoxypsoralen

5-Hydroxyxanthotoxin,5-Hydroxy-8-methoxypsoralen

5-Hydroxy-8-methoxypsoralen (5-Hydroxyxanthotoxin) is a metabolite derived from Xanthotoxin, which acts as a potent tricyclic furocoumarin suicide inhibitor of CYP (cytochrome P-450). It is employed as an agent for the treatment of psoriasis, eczema, vitiligo, and certain cutaneous Lymphomas, in combination with phototherapy involving exposure to sunlight.

天然产物

Monobenzone
Cat.No: T0759
Synonym: 4-苄氧基苯酚,Benoquin
Target: Tyrosinase
Khellin
Cat.No: T1431
Synonym: 凯林,Amicardine,Methafrone,Visammin
Target: EGFR, Others
Trioxsalen
Cat.No: T4558
Synonym: 三甲沙林,Trimethylpsoralen,Trioxysalen,Trisoralen
Target: DNA Alkylator/Crosslinker, DHFR
5-Hydroxy-8-methoxypsoralen
Cat.No: T40859
Synonym: 5-Hydroxyxanthotoxin,5-Hydroxy-8-methoxypsoralen
Target:
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