3
2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T50103 |
NFAT Inhibitor-2
|
Others | Others |
NFAT Inhibitor-2 是一种化学合成中的砌块。 | |||
T81417 |
PP5-IN-1
|
Apoptosis; Phosphatase | Apoptosis; Metabolism |
PP5-IN-1 是一种具有有效性和竞争性的丝氨酸/苏氨酸蛋白磷酸酶-5 (PP5) 抑制剂,具有潜在的抗癌活性,可诱导癌细胞凋亡。 | |||
T37056 |
D-erythro-MAPP
|
||
D-erythro-MAPP is a derivative of ceramide and an inhibitor of alkaline ceramidase (Ki = 2-13 μM; IC50 = 1-5 μM). It is selective for alkaline ceramidase over acid ceramidase (IC50 = >500 μM) as well as the serine/threonine protein phosphatase CAPP at concentrations up to 10 μM. D-erythro-MAPP increases intracellular ceramide levels, induces cell cycle arrest at the G0/G1 phase, and inhibits growth of HL-60 promyelocytic leukemia cells in a time- and concentration-dependent manner. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4915 |
β-Glycerophosphate disodium salt hydrate
|
Phosphatase; Endogenous Metabolite | Metabolism |
β-Glycerophosphate disodium salt hydrate 是一种磷酸酶抑制剂,是内源性代谢产物的一种。 | |||
T4839 |
Ac-Ala-OH
N-Acetylalanine,N-Acetyl-L-alanine,N-乙酰-L-丙氨酸 |
Others; Endogenous Metabolite | Metabolism; Others |
Ac-Ala-OH (N-Acetyl-L-alanine) 是鸟嘌呤核苷酸结合蛋白G(I)/G(S)/G(O) γ -2亚基、髓鞘碱性蛋白、GTP-结合核蛋白 Ran、原肌球蛋白 α - 4链、HIV-1 Rev 结合蛋白2、Xaa-Pro 二肽酶、胸腺酶 β -10、肌动蛋白样蛋白3、丙氨酸转氨酶、丝氨酸/苏氨酸蛋白磷酸酶PP1 - β催化亚基、10 kda 热休克蛋白(线粒体)、钙调蛋白和 β -1-syntrophin 的底物。 |