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Cat. No. Product Name Target Signaling Pathways
T36971 5-Ethynyluridine

Nucleoside Antimetabolite/Analog Cell Cycle/Checkpoint; DNA Damage/DNA Repair
5-Ethynyluridine 可用于标记新合成的 RNA。这种方法称为使用点击化学 (RICK) 捕获新转录的 RNA 相互作用组,系统地捕获与多种 RNA 结合的蛋白质,包括新生 RNA 和传统上被忽视的非多腺苷酸化 RNA。
T1046 Mexiletine hydrochloride

KOE-1173 (hydrochloride),Mexiletine HCl,KO1173,盐酸美西律

AhR; Sodium Channel Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism
Mexiletine hydrochloride (KOE-1173 hydrochloride) 是一种电压门控钠通道阻滞剂,是 IB 类抗心律失常药。 Mexiletine hydrochloride 通过抑制心肌细胞内钠电流,从而降低心脏动作电位(0相)上升速率,并且降低浦肯野纤维的自律性而发挥抗心律失常作用。
T69806 EGIS-8332

EGIS-8332 is a potent and selective non-competitive AMPA receptor antagonist. EGIS-8332 inhibits AMPA/kainate ion channels and cell death. EGIS-8332 inhibited AMPA currents in rat cerebellar Purkinje cells and inhibited the AMPA- and quisqualate-induced excitotoxicity in primary cultures of telencephalon neurons (IC(50)=5.1-9.0 microM), in vitro. EGIS-8332 seems suitable for further development for the treatment of epilepsy, ischaemia and stroke based on its efficacy in a variety of experimenta...

化合物

5-Ethynyluridine
Cat.No: T36971
Synonym:
Target: Nucleoside Antimetabolite/Analog
Mexiletine hydrochloride
Cat.No: T1046
Synonym: KOE-1173 (hydrochloride),Mexiletine HCl,KO1173,盐酸美西律
Target: AhR, Sodium Channel
EGIS-8332
Cat.No: T69806
Synonym:
Target:
TargetMol Loading
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