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Cat. No. Product Name Target Signaling Pathways
T27194 DNA Primase Inhibitor-13

DNA Primase Inhibitor-13 is a novel inhibitor of DNA primase.
T2504 Pritelivir

普瑞利韦,BAY 57-1293,AIC316

DNA/RNA Synthesis; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Pritelivir (BAY 57-1293) 是一种病毒解旋酶-引物酶复合物抑制剂,有抗病毒活性。它对 HSV-1 和 HSV-2 具有活性,IC50值为 20 nM。
T4226 Amenamevir

ASP2151,阿莫奈韦

DNA/RNA Synthesis; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Amenamevir (ASP2151) 是一种新型解旋酶引发酶抑制剂,对水痘带状疱疹病毒和 1 型和 2 型单纯疱疹病毒具有活性,EC50值为 14 ng/mL。
T6501 Fludarabine Phosphate

NSC 312887 Phosphate,fludara Phosphate,F-ara-A (NSC 312887) Phosphate,F-ara-AMP,磷酸氟达拉滨

Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Fludarabine Phosphate (NSC 312887 Phosphate) 是一种腺苷和脱氧腺苷类似物,与 dATP 竞争,并入到 DNA,可以抑制 DNA 聚合酶 α、核糖核苷酸还原酶和 DNA 引发酶,从而中断 DNA 合成并抑制肿瘤细胞生长。
T74088 Fludarabine triphosphate trisodium

Fludarabine triphosphate (F-ara-ATP) trisodium 是Fludarabine 的活性代谢物,是一种有效的、非竞争性的、特异性的DNA 引发酶 (DNA primase) 抑制剂,其IC50为 2.3 μM,Ki 为 6.1 μM。Fludarabine triphosphate trisodium 通过阻断 DNA 引发酶和引物 RNA 形成抑制 DNA 合成 (DNA synthesis)。Fludarabine triphosphate trisodium 可抑制核糖核苷酸还原酶和DNA 聚合酶,导致细胞凋亡 (apoptosis)。
T16575 Pritelivir mesylate hydrate

BAY 57-1293 mesylate hydrate,AIC316 mesylate hydrate

Others Others
Pritelivir mesylate hydrate is active against herpes simplex virus types 1 and 2 (IC50: 0.02 μM against HSV1-2). Pritelivir mesylate hydrate is an inhibitor of the viral helicase-primase complex. Pritelivir mesylate hydrate shows antiviral activity in vit
T16576 Pritelivir mesylate

BAY 57-1293 mesylate,AIC316 mesylate

Others Others
Pritelivir mesylate is active against herpes simplex virus types 1 and 2 (IC50: 0.02 μM against HSV1-2). Pritelivir mesylate is an inhibitor of the viral helicase-primase complex. Pritelivir mesylate shows antiviral activity in vitro and in animal models

化合物

DNA Primase Inhibitor-13
Cat.No: T27194
Synonym:
Target:
Pritelivir
Cat.No: T2504
Synonym: 普瑞利韦,BAY 57-1293,AIC316
Target: DNA/RNA Synthesis, HSV
Amenamevir
Cat.No: T4226
Synonym: ASP2151,阿莫奈韦
Target: DNA/RNA Synthesis, HSV
Fludarabine Phosphate
Cat.No: T6501
Synonym: NSC 312887 Phosphate,fludara Phosphate,F-ara-A (NSC 312887) Phosphate,F-ara-AMP,磷酸氟达拉滨
Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
Fludarabine triphosphate trisodium
Cat.No: T74088
Synonym:
Target:
Pritelivir mesylate hydrate
Cat.No: T16575
Synonym: BAY 57-1293 mesylate hydrate,AIC316 mesylate hydrate
Target: Others
Pritelivir mesylate
Cat.No: T16576
Synonym: BAY 57-1293 mesylate,AIC316 mesylate
Target: Others
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