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Cat. No. Product Name Target Signaling Pathways
T7587 Tenapanor

RDX-5791,RDX 5791,AZD 1722,Tenapanor free base,RDX5791,AZD-1722,AZD1722

Sodium Channel Membrane transporter/Ion channel
Tenapanor (RDX 5791) 是钠氢离子交换NHE3的有效抑制剂, 对人和大鼠NHE3的IC50分别是5和10 nM。
T6344 Sevelamer hydrochloride

Sevelamer HCl

FXR; Autophagy Autophagy; Metabolism
Sevelamer hydrochloride (Sevelamer HCl) 是一种磷酸盐结合药物,用于通过与膳食磷酸盐结合并阻止其吸收来治疗高磷血症。
T21417 Dihydrotachysterol

Hytakerol,HSDB-3314,双氢速甾醇,HSDB3314,Parterol,HSDB 3314

Dihydrotachysterol (DHT) is a biologically active synthetic analog of vitamin D. It promotes intestinal absorption of active calcium and phosphate . It is also beneficial in the treatment of hypoparathyroidism.
T70605 NaPi2b Inhibitor 15

NaPi2b is primarily expressed in the small intestine, lungs, and testes and plays an important role in phosphate homeostasis. The inhibition of NaPi2b, responsible for intestinal phosphate absorption, is considered to reduce serum phosphate levels, making it a promising therapeutic approach for hyperphosphatemia
T76151 Glycerol kinase

Glycerol kinase (GyK) 甘油激酶是一种细菌糖激酶,常用于生化研究。Glycerol kinase 通过将三醇转化为甘油-3-p (G3P) 来催化甘油代谢。Glycerol kinase 对于调节细胞中不依赖通道/促进因子的甘油摄取至关重要。

化合物

Tenapanor
Cat.No: T7587
Synonym: RDX-5791,RDX 5791,AZD 1722,Tenapanor free base,RDX5791,AZD-1722,AZD1722
Target: Sodium Channel
Sevelamer hydrochloride
Cat.No: T6344
Synonym: Sevelamer HCl
Target: FXR, Autophagy
Dihydrotachysterol
Cat.No: T21417
Synonym: Hytakerol,HSDB-3314,双氢速甾醇,HSDB3314,Parterol,HSDB 3314
Target:
NaPi2b Inhibitor 15
Cat.No: T70605
Synonym:
Target:
Glycerol kinase
Cat.No: T76151
Synonym:
Target:
TargetMol Loading
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