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Cat. No. Product Name Target Signaling Pathways
T4579 Pentagastrin

五肽胃泌素,ICI-50123

Others; cholecystokinin GPCR/G Protein; Others
Pentagastrin (ICI-50123) 是一种选择性的胆囊收缩素 B(CCKB) 受体激动剂,IC50=11 nM。它能够增强胃粘膜对酸的防御机制,并保护胃粘膜免受损伤。
T31958 Glycine-pentagastrin

Glycine pentagastrin,Boc-gly-trp-met-asp-phe-NH2,Tbgtmap

Glycine-pentagastrin can enhance gastric mucosal defence mechanisms against acid and protect the gastric mucosa from experimental injury.
T33916 Pentagastrin meglumine

Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.
T17030 Tegoprazan

ATPase; Proton pump Membrane transporter/Ion channel
Tegoprazan 是一种口服有效的、高选择性胃 H+/K+-ATP 酶 (H+/K+-ATPase) 抑制剂,能够控制胃酸分泌和运动,在体外检测的对猪、犬、人的 H+/K+-ATP 酶的 IC50为0.29-0.52 μM。
T68016 Spiroglumide

CR-2194

cholecystokinin GPCR/G Protein
Spiroglumide 是一种CCKB-胃泌素拮抗剂,能够抑制剂量依赖性五肽胃泌素诱导的酸分泌过多,其ID50为20.1(8.67-46.4)mg / kg,可用于探索胃泌素在调节人类胃酸分泌中的生理作用。
T23946 DA-3934

UNII-J353803KRG

DA-3934 has a high affinity for gastrin/CCK-B receptors and high selectivity over CCK-A receptors. DA-3934 and its methyl ester derivative inhibited pentagastrin-induced gastric acid secretion in rats in a dose-dependent manner.
T83694 Gastric Inhibitory Peptide (1-42) (porcine) TFA

GIP (1-42),Glucose-dependent Insulinotropic Polypeptide (1-42)

胃抑制肽(GIP) (1-42)是一种内源性的42氨基酸肽类肠促素激素,能诱导胰岛素分泌。该激素在肠道神经内分泌K细胞和颌下腺中表达,并在餐后释放到循环中。GIP (1-42)抑制由组胺、五肽和胰岛素引起的胃酸和胃蛋白酶分泌,增加葡萄糖诱导的胰岛素释放,并在大鼠中刺激胃排空。

化合物

Pentagastrin
Cat.No: T4579
Synonym: 五肽胃泌素,ICI-50123
Target: Others, cholecystokinin
Glycine-pentagastrin
Cat.No: T31958
Synonym: Glycine pentagastrin,Boc-gly-trp-met-asp-phe-NH2,Tbgtmap
Target:
Pentagastrin meglumine
Cat.No: T33916
Synonym:
Target:
Tegoprazan
Cat.No: T17030
Synonym:
Target: ATPase, Proton pump
Spiroglumide
Cat.No: T68016
Synonym: CR-2194
Target: cholecystokinin
DA-3934
Cat.No: T23946
Synonym: UNII-J353803KRG
Target:
Gastric Inhibitory Peptide (1-42) (porcine) TFA
Cat.No: T83694
Synonym: GIP (1-42),Glucose-dependent Insulinotropic Polypeptide (1-42)
Target:
TargetMol Loading
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