Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4579 |
Pentagastrin
五肽胃泌素,ICI-50123 |
Others; cholecystokinin | GPCR/G Protein; Others |
Pentagastrin (ICI-50123) 是一种选择性的胆囊收缩素 B(CCKB) 受体激动剂,IC50=11 nM。它能够增强胃粘膜对酸的防御机制,并保护胃粘膜免受损伤。 | |||
T31958 |
Glycine-pentagastrin
Glycine pentagastrin,Boc-gly-trp-met-asp-phe-NH2,Tbgtmap |
||
Glycine-pentagastrin can enhance gastric mucosal defence mechanisms against acid and protect the gastric mucosa from experimental injury. | |||
T33916 | Pentagastrin meglumine | ||
Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally. | |||
T17030 |
Tegoprazan
|
ATPase; Proton pump | Membrane transporter/Ion channel |
Tegoprazan 是一种口服有效的、高选择性胃 H+/K+-ATP 酶 (H+/K+-ATPase) 抑制剂,能够控制胃酸分泌和运动,在体外检测的对猪、犬、人的 H+/K+-ATP 酶的 IC50为0.29-0.52 μM。 | |||
T68016 |
Spiroglumide
CR-2194 |
cholecystokinin | GPCR/G Protein |
Spiroglumide 是一种CCKB-胃泌素拮抗剂,能够抑制剂量依赖性五肽胃泌素诱导的酸分泌过多,其ID50为20.1(8.67-46.4)mg / kg,可用于探索胃泌素在调节人类胃酸分泌中的生理作用。 | |||
T23946 |
DA-3934
UNII-J353803KRG |
||
DA-3934 has a high affinity for gastrin/CCK-B receptors and high selectivity over CCK-A receptors. DA-3934 and its methyl ester derivative inhibited pentagastrin-induced gastric acid secretion in rats in a dose-dependent manner. | |||
T83694 |
Gastric Inhibitory Peptide (1-42) (porcine) TFA
GIP (1-42),Glucose-dependent Insulinotropic Polypeptide (1-42) |
||
胃抑制肽(GIP) (1-42)是一种内源性的42氨基酸肽类肠促素激素,能诱导胰岛素分泌。该激素在肠道神经内分泌K细胞和颌下腺中表达,并在餐后释放到循环中。GIP (1-42)抑制由组胺、五肽和胰岛素引起的胃酸和胃蛋白酶分泌,增加葡萄糖诱导的胰岛素释放,并在大鼠中刺激胃排空。 |