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Cat. No.	Product Name	Target	Signaling Pathways
T2344	LY 344864 LY344864	5-HT Receptor	GPCR/G Protein; Neuroscience
	LY 344864 是一种特异性受体激动剂，有对克隆 5-HT1F 受体的亲和力，Ki 为6 nM。
T76682	Galcanezumab LY 2951742	CGRP Receptor	GPCR/G Protein; Neuroscience
	Galcanezumab 是一种靶向 CGRP 配体的人源化 IgG4 单克隆抗体，是一种与配体降钙素基因相关肽结合的抗体。Galcanezumab 可用于预防和治疗偏头痛或丛集性头痛。
T22346	Indomethacin sodium hydrate Indometacin sodium hydrate	COX	Immunology/Inflammation; Neuroscience
	Indomethacin sodium hydrate (Indometacin sodium hydrate) 是一种口服活性、竞争性和可逆性的 COX1/2 抑制剂，具有潜在的抗炎活性，可诱发的偏头痛，诱导的胃肠道损伤，可用于研究成人继发于严重创伤性脑损伤的颅内压增高和类风湿性关节。
T25616	Lanepitant 2HCl LY303870 dihydrochloride,LY 303870 dihydrochloride,LY-303870 dihydrochloride,Lanepitant dihydrochloride	Neurokinin receptor	GPCR/G Protein; Neuroscience
	Lanepitant 2HCl 是一种非肽类神经激肽-1 受体拮抗剂，具有镇痛和抗炎活性。Lanepitant 2HCl 抑制 P 物质与神经激肽-1 受体的结合，抑制神经源性炎症和疼痛传递，可用于研究偏头痛等疼痛性神经病变类疾病。
T20917	Lomerizine
	Lomerizine, a blocker of diphenylmethylpiperazine Ca2+ channel, is used to prevent migraines.
T0216L	Eletriptan UK-116,044-04 [as hydrobromide],UNII-22QOO9B8KI,UK-116,044,UK 116044
	Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.
T27196	Donitriptan Mesylate Donitriptan mesilate,F12640,F-12640,F 12640
	Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.
T70837	Rimegepant sulfate hydrate
	Rimegepant, also known as BMS-927711 and BHV-3000, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist in clinical trials for treating migraines. Rimegepant has shown in vivo efficacy without vasoconstriction effect. BMS-927711 is superior to placebo at several different doses (75 mg, 150 mg, and 300 mg) and has an excellent tolerability profile.
T26796	BI-44370
	BI-44370, a CGRP (calcitonin gene-related peptide) receptor antagonist, can be used to treat migraines and other chronic pain.
T71800	Metoprolol HCl
	Metoprolol is a selective β1 receptor blocker medication. It is used to treat high blood pressure, chest pain due to poor blood flow to the heart, and a number of conditions involving an abnormally fast heart rate. It is also used to prevent further heart problems after myocardial infarction and to prevent headaches in those with migraines.
T21558	MK-3207
	MK-3207是口服生物相容性的CGRP 受体拮抗剂，IC50和 Ki 分别为 0.12 nM 和 0.024 nM，对 AM1，AM2，CTR 和 AMY3 的抑制性较弱。MK-3207可用于偏头痛研究。