Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6713 |
Ulipristal
|
Estrogen/progestogen Receptor; Progesterone Receptor | Endocrinology/Hormones; Others |
Ulipristal 是性孕酮受体 (progesterone receptor) 的选择性调节剂。它能够与孕激素受体结合,抑制 PR 介导的基因表达,降低生殖系统中孕激素的活性。 | |||
T2527 |
Ulipristal acetate
Ulipristal,醋酸乌利司他,CDB-2914 |
Estrogen/progestogen Receptor; Progesterone Receptor; Autophagy | Autophagy; Endocrinology/Hormones; Others |
Ulipristal acetate (CDB-2914) 是一种具有抗孕酮活性的选择性孕酮受体调节剂。它可抑制子宫平滑肌瘤病的生长。它通过抑制或延迟排卵和影响子宫内膜组织,可用作紧急避孕药。 | |||
T26669 |
Asoprisnil ecamate
J956,J-956,J 956 |
||
Asoprisnil ecamate is a selective progesterone receptor modulator. Asoprisnil inhibits proliferation and induces apoptosis in cultured human uterine leiomyoma cells in the absence of comparable effects on myometrial cells. Asoprisnil inhibits embryo impla |