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4

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T6800 CCF642

AC1LYELL

Others Others
CCF642 (AC1LYELL) 是蛋白质二硫键异构酶抑制剂(IC50:2.9 μM)。它在多发性骨髓瘤细胞中引起急性内质网应激,并伴随凋亡诱导的钙释放,表现出广泛的抗多发性骨髓瘤作用。
T27417L Glutathione arsenoxide hydrochloride

GSAO HCl,Glutathione arsenoxide hydrochloride(1271726-51-2 Free base)

Apoptosis; AChR Apoptosis; Neuroscience
Glutathione arsenoxide hydrochloride (Glutathione arsenoxide hydrochloride(1271726-51-2 Free base)) 是一种潜在的抗癌活性分子和肿瘤代谢抑制剂。Glutathione arsenoxide hydrochloride 靶向线粒体内膜腺嘌呤核苷酸转移酶 (ANT),对细胞增殖有抑制作用,促进细胞凋亡。Glutathione arsenoxide hydrochloride 可用于识别如蛋白质二硫异构酶一样的细胞表面蛋白质。
T19260 D-Erythrose 4-phosphate sodium

Others Others
D-erythrose 4-sodium phosphate is the sodium phosphate of the monosaccharide erythrose. Erythritol is actually converted to D-erythrose 4-phosphate involving three isomerases.
T38115 Fluprostenol serinol amide

2-arachidonyl glycerol (2-AG) exhibits cannabinoid (CB) agonist activity at the CB1 receptor, is an important endogenous monoglyceride species, and is thus considered to be the natural ligand for the CB1 receptor. 2-AG can also be metabolized by cyclooxygenase-2 and specific prostaglandin H2 (PGH2) isomerases to form PG 2-glyceryl esters. Fluprostenol serinol amide (Flu-SA) is a stable analog of PGF2α 2-glyceryl ester that has much greater stability. The biological activity of Flu-SA has not yet...

化合物

CCF642
Cat.No: T6800
Synonym: AC1LYELL
Target: Others
Glutathione arsenoxide hydrochloride
Cat.No: T27417L
Synonym: GSAO HCl,Glutathione arsenoxide hydrochloride(1271726-51-2 Free base)
Target: Apoptosis, AChR
D-Erythrose 4-phosphate sodium
Cat.No: T19260
Synonym:
Target: Others
Fluprostenol serinol amide
Cat.No: T38115
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0588 D-(-)-Arabinose

D-阿拉伯糖,D(-)-Arabinose,D-arabinose

Others Others
D-(-)-Arabinose 是一种单糖,对秀丽隐杆线虫有较强的生长抑制作用(IC50:7.5 mM)。
T4010 Juglone

5-羟基对萘醌,5-Hydroxy-1,4-naphthoquinone,胡桃酮,Regianin

DNA/RNA Synthesis; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Juglone (Regianin) 是一种从黑胡桃Juglans regia 中发现的黄色染料,有抗菌作用。

天然产物

D-(-)-Arabinose
Cat.No: T0588
Synonym: D-阿拉伯糖,D(-)-Arabinose,D-arabinose
Target: Others
Juglone
Cat.No: T4010
Synonym: 5-羟基对萘醌,5-Hydroxy-1,4-naphthoquinone,胡桃酮,Regianin
Target: DNA/RNA Synthesis, Antibacterial
TargetMol Loading
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