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Cat. No. Product Name Target Signaling Pathways
T15207 Eleclazine hydrochloride

GS 6615 hydrochloride

Sodium Channel Membrane transporter/Ion channel
Eleclazine hydrochloride (GS 6615 hydrochloride) 是新型 Na+电流抑制剂,IC50是0.7 uM。
T75098 HIF-PHD-IN-3

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
HIF-PHD-IN-3 是一种有效的 hiPSC-CM 心脏保护支架,对 HIF-PHD 有潜在的抑制作用,可调节血红素加氧酶-1,可用于研究贫血。
T27064 CP-312

CP312,Cardioprotectant 312

Reactive Oxygen Species; Autophagy Autophagy; Immunology/Inflammation; Metabolism; NF-κB
CP-312 (Cardioprotectant 312)是一种抗氧化防御反应激活剂,它通过诱导血红素加氧酶-1发挥作用,通过诱导 HMOX1 表达来靶向抗氧化反应网络,从而保护 hiPSC-CM 的活力。CP-312 保护人 iPSC 衍生的心肌细胞免受氧化应激。
T79208 Oct4 inducer-2

Oct4 inducer-2, 作为OCT4诱导剂,维持hiPSC形成通过促进内源性OCT4表达,适用于抗衰老研究。
T68485 Apilimod HCl

Apilimod dimesylate is a potent and selective PIKfyve inhibitor. It exhibits no significant activity at other lipid kinases and protein kinases, including PIP4K, PIP5K, mTOR, PI3K and PI4K. Apilimod dimesylate inhibits cellular entry by SARS-CoV-2, MERS-CoV and MHV S pseudovirions. It reduces the number of SARS-CoV-2-infected hiPSC-derived pneumocyte-like cells by 85% and inhibits SARS-CoV-2 replication in donor lung tissue. It also exhibits selective cytotoxicity in B-cell non-Hodgkin lymphoma ...

化合物

Eleclazine hydrochloride
Cat.No: T15207
Synonym: GS 6615 hydrochloride
Target: Sodium Channel
HIF-PHD-IN-3
Cat.No: T75098
Synonym:
Target: Reactive Oxygen Species
CP-312
Cat.No: T27064
Synonym: CP312,Cardioprotectant 312
Target: Reactive Oxygen Species, Autophagy
Oct4 inducer-2
Cat.No: T79208
Synonym:
Target:
Apilimod HCl
Cat.No: T68485
Synonym:
Target:
TargetMol Loading
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