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Cat. No. Product Name Target Signaling Pathways
T15159 Dorzagliatin

HMS5552

Glucokinase Metabolism
Dorzagliatin (HMS5552) 是双重作用的葡萄糖激酶 (glucokinase;GK) 激活剂,可改善 2 型糖尿病的血糖控制,提高胰腺 β 细胞功能。
T62656 GPR81 agonist 1

GPR Endocrinology/Hormones; GPCR/G Protein
GPR81 agonist 1 是一种具有高效性和选择性的 GPR81 激动剂,对人和小鼠 GPR81 具有很高的亲和力。GPR81 agonist 1 抑制分化的 3T3-L1 脂肪细胞的脂解,改善胰岛素抵抗和糖尿病小鼠模型的胰岛素敏感性和血糖控制,可用于研究糖尿病和肥胖。
TP1566 GIP (1-30) amide (Human) (TFA)

GIP (1-30) amide (Human) TFA is a glucose-dependent insulinotropic polypeptide fragment. Glucose-dependent insulinotropic polypeptide (GIP) is an incretin hormone that stimulates insulin secretion and reduces postprandial glycaemic excursions.
T64475 FMOC-L-THR

FMOC-L-THR (AZP-531) is an analogue of unacylated ghrelin designed to improve glycaemic control and reduce weight. The O-glycosidic linkage and the O-acetyl protection in this building block is stable to both piperidine and TFA, making it completely compatible with standard protocols in Fmoc solid phase peptide synthesis. The Tn antigen is a tumor-associated carbohydrate antigen that is not normally expressed in peripheral tissues or blood cells. Expression of this antigen, which is found in a m...

化合物

Dorzagliatin
Cat.No: T15159
Synonym: HMS5552
Target: Glucokinase
GPR81 agonist 1
Cat.No: T62656
Synonym:
Target: GPR
GIP (1-30) amide (Human) (TFA)
Cat.No: TP1566
Synonym:
Target:
FMOC-L-THR
Cat.No: T64475
Synonym:
Target:
TargetMol Loading
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