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Cat. No. Product Name Target Signaling Pathways
T1069 Metoclopramide hydrochloride

盐酸甲氧氯普胺,Maxolon,Metoclopramide HCl

Dopamine Receptor; 5-HT Receptor; AChR GPCR/G Protein; Neuroscience
Metoclopramide hydrochloride (Metoclopramide HCl) 是可口服的5-HT3和多巴胺D2受体拮抗剂,IC50值分别为 308 和 483 nM,用于恶心呕吐、胃食管反流和胃轻瘫的研究。
T4616 Metoclopramide

甲氧氯普胺,胃复安,5-Chloro-2-methoxyprocainamide

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Metoclopramide (5-Chloro-2-methoxyprocainamide) 是5-HT3和多巴胺D2受体拮抗剂,IC50值分别为 308 和 483 nM,可用于恶心呕吐、胃食管反流和胃轻瘫的研究。
T8385 Metoclopramide hydrochloride hydrate

盐酸甲氧氯普胺,甲氧氯普胺盐酸水合物,Metoclopramide monohydrochloride monohydrate

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) 是5-HT3和多巴胺D2受体拮抗剂,IC50值分别为 308 和 483 nM,可用于恶心呕吐、胃食管反流和胃轻瘫的研究。
T38754 Trazpiroben

TAK-906

Dopamine Receptor GPCR/G Protein; Neuroscience
Trazpiroben (TAK-906) 是一种选择性多巴胺 D2/D3 受体拮抗剂,用于研究胃痉挛。
TP2403 Recanaclotide

IW 9179,IW-9179,IW9179

Recanaclotide can be used to treat Gastroparesis, Functional Dyspepsia, and Other Gastrointestinal Disorders.
T71632 TZP-102

TZP-102 is a potent, oral, ghrelin receptor agonist that has been shown to improve diabetic gastroparesis symptoms.
T35046 Velusetrag

TD 5108,TD5108,TD-5108

Velusetrag(TD-5108)is an effective, selective, and highly potent agonist of the 5-HT4 receptor, and being developed for the treatment of gastroparesis, chronic constipation, and irritable bowel syndrome.
T62973 DS-3801b

DS-3801b 是一种强效的、非大环内酯类 GPR38 激动剂。DS-3801b 具有潜力成为研究功能性胃肠道疾病(如胃痉挛、慢性便秘)的新型胃肠道促动剂。
T39236 Relamorelin acetate

Relamorelin acetate,RM-131 acetate,BIM-28131acetate

Relamorelin (RM-131) acetate is a pentapeptide ghrelin analog that acts as a selective agonist for the ghrelin/growth hormone secretagogue receptor (GHSR). It exhibits a high affinity for the GHS-1a receptor, with a Ki value of 0.42 nM. Notably, Relamorelin acetate can cross the blood-brain barrier and target the central nervous system. This compound effectively increases growth hormone levels and promotes faster gastric emptying. Due to these properties, Relamorelin acetate holds promise for it...
T75262 Relamorelin TFA

Relamorelin (RM-131) TFA,一种生长素类似物,是一种选择性的生长素释放肽/生长激素促分泌素受体 (GHSR) 激动剂,对GHS-1a 受体的Ki 值为 0.42 nM。Relamorelin TFA 是一种五肽,具有中枢渗透性。Relamorelin TFA 增加生长激素水平,加速胃排空,具有用于恶病质、胃轻瘫和胃/肠运动障碍研究的潜力。

化合物

Metoclopramide hydrochloride
Cat.No: T1069
Synonym: 盐酸甲氧氯普胺,Maxolon,Metoclopramide HCl
Target: Dopamine Receptor, 5-HT Receptor, AChR
Metoclopramide
Cat.No: T4616
Synonym: 甲氧氯普胺,胃复安,5-Chloro-2-methoxyprocainamide
Target: Dopamine Receptor, 5-HT Receptor
Metoclopramide hydrochloride hydrate
Cat.No: T8385
Synonym: 盐酸甲氧氯普胺,甲氧氯普胺盐酸水合物,Metoclopramide monohydrochloride monohydrate
Target: Dopamine Receptor, 5-HT Receptor
Trazpiroben
Cat.No: T38754
Synonym: TAK-906
Target: Dopamine Receptor
Recanaclotide
Cat.No: TP2403
Synonym: IW 9179,IW-9179,IW9179
Target:
TZP-102
Cat.No: T71632
Synonym:
Target:
Velusetrag
Cat.No: T35046
Synonym: TD 5108,TD5108,TD-5108
Target:
DS-3801b
Cat.No: T62973
Synonym:
Target:
Relamorelin acetate
Cat.No: T39236
Synonym: Relamorelin acetate,RM-131 acetate,BIM-28131acetate
Target:
Relamorelin TFA
Cat.No: T75262
Synonym:
Target:
TargetMol Loading
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