Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T66866 | 4-Ethyl-5-fluoropyrimidine | ||
4-Ethyl-5-fluoropyrimidine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66866,CAS号为 137234-88-9。 | |||
T7718 |
5-Fluoro-2'-deoxycytidine
5-氟脱氧胞苷,FdCyd,2'-DEOXY-5-FLUOROCYTIDINE |
DNA Methyltransferase | Chromatin/Epigenetic |
5-Fluoro-2'-deoxycytidine (2'-DEOXY-5-FLUOROCYTIDINE) 是一种 DNA 甲基转移酶(DNMT) 抑制剂,是氟嘧啶核苷类似物。它是胸苷酸合酶抑制剂 5-fluoro-2′-dUMP 的肿瘤选择性前药。 | |||
T1600 |
Doxifluridine
Ro 21-9738,AMC 0101,5'-DFUR,5-Fluoro-5'-deoxyuridine,去氧氟尿苷 |
Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Doxifluridine (AMC 0101) 是一种胸苷磷酸化酶活化剂,对 PC9-DPE2细胞的 IC50为0.62 μM。它是具有抗肿瘤活性的抗肿瘤剂 5-fluorouracil (5-FU) 的氟嘧啶衍生物和口服前药。 | |||
T1408 |
Capecitabine
Xeloda,卡培他滨,Capecitibine,Capiibine,RO 09-1978 |
Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Capecitabine (Capecitibine) 是一种可口服的前药,可由胸苷磷酸化酶催化转变为其活性代谢物 Fluorouracil。 | |||
T13089 |
TAS-114
|
Others | Others |
TAS-114 is a dual inhibitor of dUTPase/dihydropyrimidine dehydrogenase (DPD), and can improving the therapeutic efficacy of fluoropyrimidine. |