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Cat. No. Product Name Target Signaling Pathways
T66866 4-Ethyl-5-fluoropyrimidine

4-Ethyl-5-fluoropyrimidine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66866,CAS号为 137234-88-9。
T7718 5-Fluoro-2'-deoxycytidine

5-氟脱氧胞苷,FdCyd,2'-DEOXY-5-FLUOROCYTIDINE

DNA Methyltransferase Chromatin/Epigenetic
5-Fluoro-2'-deoxycytidine (2'-DEOXY-5-FLUOROCYTIDINE) 是一种 DNA 甲基转移酶(DNMT) 抑制剂,是氟嘧啶核苷类似物。它是胸苷酸合酶抑制剂 5-fluoro-2′-dUMP 的肿瘤选择性前药。
T1600 Doxifluridine

Ro 21-9738,AMC 0101,5'-DFUR,5-Fluoro-5'-deoxyuridine,去氧氟尿苷

Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Doxifluridine (AMC 0101) 是一种胸苷磷酸化酶活化剂,对 PC9-DPE2细胞的 IC50为0.62 μM。它是具有抗肿瘤活性的抗肿瘤剂 5-fluorouracil (5-FU) 的氟嘧啶衍生物和口服前药。
T1408 Capecitabine

Xeloda,卡培他滨,Capecitibine,Capiibine,RO 09-1978

Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Capecitabine (Capecitibine) 是一种可口服的前药,可由胸苷磷酸化酶催化转变为其活性代谢物 Fluorouracil。
T13089 TAS-114

Others Others
TAS-114 is a dual inhibitor of dUTPase/dihydropyrimidine dehydrogenase (DPD), and can improving the therapeutic efficacy of fluoropyrimidine.

化合物

4-Ethyl-5-fluoropyrimidine
Cat.No: T66866
Synonym:
Target:
5-Fluoro-2'-deoxycytidine
Cat.No: T7718
Synonym: 5-氟脱氧胞苷,FdCyd,2'-DEOXY-5-FLUOROCYTIDINE
Target: DNA Methyltransferase
Doxifluridine
Cat.No: T1600
Synonym: Ro 21-9738,AMC 0101,5'-DFUR,5-Fluoro-5'-deoxyuridine,去氧氟尿苷
Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
Capecitabine
Cat.No: T1408
Synonym: Xeloda,卡培他滨,Capecitibine,Capiibine,RO 09-1978
Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
TAS-114
Cat.No: T13089
Synonym:
Target: Others
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