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Search Results for " fibrillogenesis "

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抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0382 Eprodisate disodium

NC-503,伊罗地塞二钠,伊罗地塞二钠盐

Others Others
Eprodisate disodium (NC-503) 是一种带负电荷的磺化类的原纤维形成抑制剂,是口服具有活力的 Eprodisate 二钠盐形式,可用于研究淀粉样蛋白A(AA) 淀粉样变性病。
T11207 Entacapone sodium salt

Others Others
Entacapone sodium salt inhibits catechol-O-methyltransferase(COMT) with similar IC50 in different tissues including live, duodenum, kidney and lung, but entacapone is more active than tolcapone in those tissues. Entacapone (< 100 μM) is a potent inhibitor of α-syn and β-amyloid (Aβ) oligomerization and fibrillogenesis, and also protects against extracellular toxicity induced by the aggregation of both proteins in PC12 cells.Entacapone sodium salt is a specific, potent, peripherally acting catech...
T80104 Z-Phe-Ala-diazomethylketone

PADK

Z-Phe-Ala-diazomethylketone 直接与 Aβ42 单体及其小型低聚物相结合,能抑制 Aβ42 在溶液中形成的十二聚体以及原纤维的生成,显示出在神经退行性疾病研究中的应用潜力。

化合物

Eprodisate disodium
Cat.No: T0382
Synonym: NC-503,伊罗地塞二钠,伊罗地塞二钠盐
Target: Others
Entacapone sodium salt
Cat.No: T11207
Synonym:
Target: Others
Z-Phe-Ala-diazomethylketone
Cat.No: T80104
Synonym: PADK
Target:
Cat. No. Product Name Target Signaling Pathways
T1686 Hematoxylin

苏木精,Hydroxybrazilin,Natural Black 1,Haematoxylin

Beta Amyloid; Others Neuroscience; Others
Hematoxylin (Natural Black 1) 是一种天然存在的类黄酮化合物,衍生自木柴树Haematoxylon campechianum。它是一种组织学上的核染色剂,也是一种有效的Aβ42原纤维形成的抑制剂,IC50=1.6 µM。
TN1216 2-O-Acetyl-20-hydroxyecdysone

20-Hydroxyeedysone 2-acetate

Beta Amyloid; Others Neuroscience; Others
2-O-Acetyl-20-hydroxyecdysone 是存在于昆虫和陆生植物中的一种蜕皮激素,2-O-Acetyl-20-hydroxyecdysone 对 amyloid-β42 诱导的细胞毒性有抑制作用,能够通过促进纤维发生减少 Aβ 寡聚物的形成,将 Aβ 寡聚物转变为低毒性纤维。

天然产物

Hematoxylin
Cat.No: T1686
Synonym: 苏木精,Hydroxybrazilin,Natural Black 1,Haematoxylin
Target: Beta Amyloid, Others
2-O-Acetyl-20-hydroxyecdysone
Cat.No: TN1216
Synonym: 20-Hydroxyeedysone 2-acetate
Target: Beta Amyloid, Others
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