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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T22459 Xanthinol Nicotinate

Angioamin,烟酸占替诺,Complamin

Others Others
Xanthinol Nicotinate (Complamin) 是血管扩张剂,可直接作用于小动脉和毛细血管的平滑肌,能够扩大血管,改善血液流变学并降低外周血管阻力。
T1115 Doxylamine succinate

琥珀酸多西拉敏,Decapryn

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Doxylamine succinate (Decapryn) 是一种吡啶衍生物组胺 H1 拮抗剂,具有明显的镇静特性。它竞争性阻断组胺 H1 受体并限制典型的过敏和过敏反应,可防止组胺引起的皮肤和粘膜疼痛和瘙痒。
T21020 Antazoline phosphate

Antazoline phosphate is an antihistamine with anticholinergic properties. Antazoline prevents the typical allergic symptoms on capillaries, mucous membranes, skin, and gastrointestinal and bronchial smooth muscles by antagonizing the histamine H1 receptor
T70129 ST-115

ST-115 is a potent and specific inhibitor of aminopeptidase P2. When ST-115 is administered intravenously at the start of reperfusion, it reduces bradykinin degradation. This increases bradykinin's concentration in the capillaries and enhances its protective effects.

化合物

Xanthinol Nicotinate
Cat.No: T22459
Synonym: Angioamin,烟酸占替诺,Complamin
Target: Others
Doxylamine succinate
Cat.No: T1115
Synonym: 琥珀酸多西拉敏,Decapryn
Target: Histamine Receptor
Antazoline phosphate
Cat.No: T21020
Synonym:
Target:
ST-115
Cat.No: T70129
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2520 Desloratadine

Sch34117,地氯雷他定,NSC 675447

Endogenous Metabolite; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Desloratadine (Sch34117) 是非镇静H1抗组胺药 Loratadine 的主要口服代谢物,可减少对支气管平滑肌、毛细血管和胃肠道平滑肌中 H1 受体的典型组胺能作用,包括血管舒张、支气管收缩、血管通透性增加、疼痛、瘙痒和胃肠道平滑肌的痉挛性收缩。它是一种选择性H1受体拮抗剂,具有抗过敏和抗炎活性。
T6535 Histamine Phosphate

组胺磷酸盐,Histamine diphosphate,二磷酸组胺,Histamine acid phosphate

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Histamine Phosphate (Histamine acid phosphate) 是组胺受体的强激活剂和血管扩张神经剂,可激活一氧化氮合成酶。

天然产物

Desloratadine
Cat.No: T2520
Synonym: Sch34117,地氯雷他定,NSC 675447
Target: Endogenous Metabolite, Histamine Receptor
Histamine Phosphate
Cat.No: T6535
Synonym: 组胺磷酸盐,Histamine diphosphate,二磷酸组胺,Histamine acid phosphate
Target: Histamine Receptor
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