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5
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T62091 |
Anti-hyperglycemic agent-1
|
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Anti-hyperglycemic agent 1 是一种 α- 葡萄糖苷酶 (α-Glucosidase) 的有效抑制剂 (IC50: 0.53 μM)。Anti-hyperglycemic agent 1 能够用于研究糖尿病。 | |||
T32754 |
Limiglidole
|
||
Limiglidole is an anti-hyperglycemic drug candidate. | |||
T10362L |
AR453588 hydrochloride
|
Others | Others |
AR453588 hydrochloride is an orally bioavailable anti-diabetic glucokinase activator (EC50: 42 nM) with anti-hyperglycemic activity. | |||
T30166 |
ASP-4000 HCl
ASP4000 HCl,ASP 4000 HCl,UNII-7393JFE67B |
||
ASP-4000 HCl is an inhibitor of dipeptidyl peptidase 4 (DPP) with anti-hyperglycemic activity. | |||
T10362 |
AR453588
|
Others | Others |
AR453588 is an orally bioavailable anti-diabetic glucokinase activator (EC50: 42 nM) with anti-hyperglycemic activity. | |||
T80715 | α-Amylase/α-Glucosidase-IN-6 | ||
α-Amylase/α-Glucosidase-IN-6 (compound 5j) 是一种对α-amylase和α-glucosidase具有双重抑制作用的有效化合物,其IC50s分别为17.0 µM和40.1 µM。该化合物还表现出抗高血糖活性。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3672 |
Nomilin
|
MAPK | MAPK |
Nomilin 是一种柠檬苦素类化合物,从柑桔类提取物中获得,是抗肥胖症和降糖药。 | |||
TN1513 |
Clitorin
碟豆宁,碟豆素 |
PKC; Antifection | Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology |
Clitorin 是一种山奈酚糖苷,分离自 Acalypha indica 的花和叶,表现出抗氧化活性。 | |||
TN6793 |
Demethylisoencecalin
6-Acetyl-5-hydroxy-2,2-dimethyl-2H-1-benzopyran |
Others | Others |
Demethylisoencecalin (6-Acetyl-5-hydroxy-2,2-dimethyl-2H-1-benzopyran) 具有抗高血糖活性。 | |||
T3747 |
syringaldehyde
Syringic aldehyde,丁香醛,Springaldehyde |
COX | Immunology/Inflammation; Neuroscience |
syringaldehyde 是可从厚朴和木薯中分离得到的黄酮类多酚,具有抗氧化、抗高血糖和抗炎活性,可适度抑制COX-2活性,IC50为 3.5 μg/mL。 | |||
TN3532 | Borapetoside E | Others | Others |
Borapetoside E has anti-hyperglycemic activity, it can significantly reduce serum glucose levels at dose-dependent manners in alloxan-induced hyperglycemic mice and db/db type 2 diabetic mice. |