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Search Results for " anti-hyperglycemic "

6

抑制剂 & 化合物

5

天然产物

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Cat. No. Product Name Target Signaling Pathways
T62091 Anti-hyperglycemic agent-1

Anti-hyperglycemic agent 1 是一种 α- 葡萄糖苷酶 (α-Glucosidase) 的有效抑制剂 (IC50: 0.53 μM)。Anti-hyperglycemic agent 1 能够用于研究糖尿病。
T32754 Limiglidole

Limiglidole is an anti-hyperglycemic drug candidate.
T10362L AR453588 hydrochloride

Others Others
AR453588 hydrochloride is an orally bioavailable anti-diabetic glucokinase activator (EC50: 42 nM) with anti-hyperglycemic activity.
T30166 ASP-4000 HCl

ASP4000 HCl,ASP 4000 HCl,UNII-7393JFE67B

ASP-4000 HCl is an inhibitor of dipeptidyl peptidase 4 (DPP) with anti-hyperglycemic activity.
T10362 AR453588

Others Others
AR453588 is an orally bioavailable anti-diabetic glucokinase activator (EC50: 42 nM) with anti-hyperglycemic activity.
T80715 α-Amylase/α-Glucosidase-IN-6

α-Amylase/α-Glucosidase-IN-6 (compound 5j) 是一种对α-amylase和α-glucosidase具有双重抑制作用的有效化合物,其IC50s分别为17.0 µM和40.1 µM。该化合物还表现出抗高血糖活性。

化合物

Anti-hyperglycemic agent-1
Cat.No: T62091
Synonym:
Target:
Limiglidole
Cat.No: T32754
Synonym:
Target:
AR453588 hydrochloride
Cat.No: T10362L
Synonym:
Target: Others
ASP-4000 HCl
Cat.No: T30166
Synonym: ASP4000 HCl,ASP 4000 HCl,UNII-7393JFE67B
Target:
AR453588
Cat.No: T10362
Synonym:
Target: Others
α-Amylase/α-Glucosidase-IN-6
Cat.No: T80715
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3672 Nomilin

MAPK MAPK
Nomilin 是一种柠檬苦素类化合物,从柑桔类提取物中获得,是抗肥胖症和降糖药。
TN1513 Clitorin

碟豆宁,碟豆素

PKC; Antifection Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology
Clitorin 是一种山奈酚糖苷,分离自 Acalypha indica 的花和叶,表现出抗氧化活性。
TN6793 Demethylisoencecalin

6-Acetyl-5-hydroxy-2,2-dimethyl-2H-1-benzopyran

Others Others
Demethylisoencecalin (6-Acetyl-5-hydroxy-2,2-dimethyl-2H-1-benzopyran) 具有抗高血糖活性。
T3747 syringaldehyde

Syringic aldehyde,丁香醛,Springaldehyde

COX Immunology/Inflammation; Neuroscience
syringaldehyde 是可从厚朴和木薯中分离得到的黄酮类多酚,具有抗氧化、抗高血糖和抗炎活性,可适度抑制COX-2活性,IC50为 3.5 μg/mL。
TN3532 Borapetoside E

Others Others
Borapetoside E has anti-hyperglycemic activity, it can significantly reduce serum glucose levels at dose-dependent manners in alloxan-induced hyperglycemic mice and db/db type 2 diabetic mice.

天然产物

Nomilin
Cat.No: T3672
Synonym:
Target: MAPK
Clitorin
Cat.No: TN1513
Synonym: 碟豆宁,碟豆素
Target: PKC, Antifection
Demethylisoencecalin
Cat.No: TN6793
Synonym: 6-Acetyl-5-hydroxy-2,2-dimethyl-2H-1-benzopyran
Target: Others
syringaldehyde
Cat.No: T3747
Synonym: Syringic aldehyde,丁香醛,Springaldehyde
Target: COX
Borapetoside E
Cat.No: TN3532
Synonym:
Target: Others
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