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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1199 |
Mitotane
Mitotan,o,p'-DDD,NCI-C04933,2,4′-DDD,米托坦 |
Apoptosis; AChR | Apoptosis; Neuroscience |
Mitotane (NCI-C04933) 是 DDD 的同分异构体和 DDT 的衍生物,可作用于肾上腺皮质癌,有抗癌活性。 | |||
T8401 |
Efonidipine hydrochloride monoethanolate
NZ-105 hydrochloride monoethanolate,依福地平,盐酸依福地平一乙醇盐 |
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Efonidipine hydrochloride monoethanolate (NZ-105 hydrochloride monoethanolate) 是 T 型和 L 型钙离子通道双重阻断剂。 | |||
T19737 | Perthane | ||
Perthane is the diethyl derivative of common pesticide DDD. It may cause adrenocortical atrophy in humans,and also prevent the formation of spontaneous mammary carcinoma. | |||
T75135 | FHD-609 | ||
FHD-609 为含溴结构域蛋白BRD9的抑制剂及降解剂,针对ncBAF,适用于研究含BAF复合亚基突变的多种癌症。FHD-609与Telomelysin或INO5401联用,或对肾上腺皮质癌(ACC)的研究具有潜在作用。 | |||
T72213 |
Efonidipine hydrochloride
NZ-105 hydrochloride |
||
Efonidipine(NZ-105)盐酸盐是T 型和L 型钙离子通道双重阻断剂。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T36472 |
Tetrahydro-11-deoxy Cortisol
|
||
Tetrahydro-11-deoxy cortisol (THS) is the primary urinary metabolite of 11-deoxycortisol. Urinary excretion of THS is elevated in patients with 11β-hydroxylase deficiency, a condition resulting from mutations in the cytochrome P450 (CYP) isoform CYP11B1. Urinary levels of THS are also elevated in patients with adrenocortical carcinoma (ACC) and adrenocortical adenoma (ACA) but are higher in patients with ACC compared to ACA. |