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Search Results for " adrenocortical carcinoma "

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抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T1199 Mitotane

Mitotan,o,p'-DDD,NCI-C04933,2,4′-DDD,米托坦

Apoptosis; AChR Apoptosis; Neuroscience
Mitotane (NCI-C04933) 是 DDD 的同分异构体和 DDT 的衍生物,可作用于肾上腺皮质癌,有抗癌活性。
T8401 Efonidipine hydrochloride monoethanolate

NZ-105 hydrochloride monoethanolate,依福地平,盐酸依福地平一乙醇盐

Calcium Channel Membrane transporter/Ion channel; Metabolism
Efonidipine hydrochloride monoethanolate (NZ-105 hydrochloride monoethanolate) 是 T 型和 L 型钙离子通道双重阻断剂。
T19737 Perthane

Perthane is the diethyl derivative of common pesticide DDD. It may cause adrenocortical atrophy in humans,and also prevent the formation of spontaneous mammary carcinoma.
T75135 FHD-609

FHD-609 为含溴结构域蛋白BRD9的抑制剂及降解剂,针对ncBAF,适用于研究含BAF复合亚基突变的多种癌症。FHD-609与Telomelysin或INO5401联用,或对肾上腺皮质癌(ACC)的研究具有潜在作用。
T72213 Efonidipine hydrochloride

NZ-105 hydrochloride

Efonidipine(NZ-105)盐酸盐是T 型和L 型钙离子通道双重阻断剂。

化合物

Mitotane
Cat.No: T1199
Synonym: Mitotan,o,p'-DDD,NCI-C04933,2,4′-DDD,米托坦
Target: Apoptosis, AChR
Efonidipine hydrochloride monoethanolate
Cat.No: T8401
Synonym: NZ-105 hydrochloride monoethanolate,依福地平,盐酸依福地平一乙醇盐
Target: Calcium Channel
Perthane
Cat.No: T19737
Synonym:
Target:
FHD-609
Cat.No: T75135
Synonym:
Target:
Efonidipine hydrochloride
Cat.No: T72213
Synonym: NZ-105 hydrochloride
Target:
Cat. No. Product Name Target Signaling Pathways
T36472 Tetrahydro-11-deoxy Cortisol

Tetrahydro-11-deoxy cortisol (THS) is the primary urinary metabolite of 11-deoxycortisol. Urinary excretion of THS is elevated in patients with 11β-hydroxylase deficiency, a condition resulting from mutations in the cytochrome P450 (CYP) isoform CYP11B1. Urinary levels of THS are also elevated in patients with adrenocortical carcinoma (ACC) and adrenocortical adenoma (ACA) but are higher in patients with ACC compared to ACA.

天然产物

Tetrahydro-11-deoxy Cortisol
Cat.No: T36472
Synonym:
Target:
TargetMol Loading
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