Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7704 |
KY-226
|
Phosphatase | Metabolism |
KY-226 是选择性的,口服活性的和变构蛋白酪氨酸磷酸酶 1B 抑制剂,IC50=0.25 μM,且不激活 PPARγ 。它可以保护神经元免受脑缺血损伤。它通过增强胰岛素和瘦素信号传导发挥抗糖尿病和抗肥胖作用。 | |||
T16684 |
Puromycin aminonucleoside
维生素E醋酸酯,NSC 3056 |
Apoptosis; Proteasome; Aminopeptidase; Antibacterial; Antibiotic | Apoptosis; Metabolism; Microbiology/Virology; Proteases/Proteasome; Ubiquitination |
Puromycin aminonucleoside (NSC-3056) 是一种氨基核苷类抗生素,是嘌呤霉素类似物。它可逆抑制二肽基肽酶和胞浆丙氨酸氨基肽酶。它通过以氧化应激依赖性方式调节 ZO-1 来增加足细胞通透性。它诱导细胞凋亡 。 | |||
T70232 | 3,4-Dephostatin | ||
3,4-Dephostatin is an inhibitor of the interactions of CFTR-associated ligand (CAL) and PSD-95/Dlg1/ZO-1 (PDZ) domain. | |||
T69658 | Ethyl-3,4-dephostatin | ||
Ethyl-3,4-dephostatin is a novel inhibitor of the interactions of CFTR-associated ligand and PSD-95/Dlg1/ZO-1 domain. |