Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1846 |
Y-320
Y320 |
IL Receptor; Lipase; Interleukin | Immunology/Inflammation; Metabolism |
Y-320 是一种免疫调节剂,能阻碍IL-15刺激CD4 T 细胞后的IL-17的产生,IC50=20~60 nM。 | |||
T5125 |
LY3200882
|
TGF-beta/Smad | Stem Cells |
LY3200882 是一种高度选择性的、口服活性的、具有 ATP 竞争性的 TGF-β 受体 1 型 (ALK5) 抑制剂(IC50:38.2 nM)。它能够抑制多种促肿瘤活性,可用作免疫调节剂。 | |||
T27944 |
LY3202626
LY 3202626,LY-3202626 |
||
LY3202626, an amyloid precursor protein secretase (BACE protein) inhibitor, is used for the treatment of Alzheimer's disease. | |||
T22951 |
LY320135
LY 320135 |
Others | Others |
CB1 receptor antagonist/inverse agonist | |||
T27945 |
LY320954
LY 320954,PDSP1_001629,LY-320954 |
||
LY320954 is an antagonist of 5-HT2A receptor. |